SCHEMBL2833139

SCHEMBL2833139

CCCc1c(C)nn(-c2c(Cl)cccc2Cl)c1COc1ccc(-c2ccc(C(=O)O)cc2)c(C)c1

nearest known ligand 0.44

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
NR1H4 Q96RI1 9/20 0.44
MRGPRX4 Q96LA9 1/20 0.41
NR4A2 P43354 2/20 0.39
PTPN11 Q06124 1/20 0.39
RXRA P19793 1/20 0.38
RXRB P28702 1/20 0.38
RXRG P48443 1/20 0.38
RARB P10826 1/20 0.38
NPC1 O15118 1/20 0.37
RAB9A P51151 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2773781 0.93 NR1H4 (0.45) NR1H4MRGPRX4NR4A2PTPN11RXRA
SCHEMBL2773617 0.89 NR1H4 (0.47) NR1H4MRGPRX4NR4A2
SCHEMBL2772558 0.88 NR1H4 (0.47) NR1H4MRGPRX4NR4A2RXRARXRB
SCHEMBL2772065 0.85 NR1H4 (0.46) NR1H4MRGPRX4NR4A2RXRARXRB
SCHEMBL2772063 0.84 PPARA (0.43) NR1H4MRGPRX4NR4A2RXRARXRB
SCHEMBL2774437 0.83 NR1H4 (0.50) NR1H4MRGPRX4NR4A2RXRARXRB
SCHEMBL2771298 0.81 NR1H4 (0.60) NR1H4
SCHEMBL2775206 0.81 MRGPRX4 (0.48) NR1H4MRGPRX4
SCHEMBL2771295 0.81 NR1H4 (0.60) NR1H4
SCHEMBL3150343 0.80 NR1H4 (0.51) NR1H4MRGPRX4NR4A2PTPN11

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2029547-B1 FXR AGONISTS LILLY CO ELI (US) 2010-04-28 EP disclosed