SCHEMBL27745441

SCHEMBL27745441

Cn1nc2ccccc2c1C(=O)NN

nearest known ligand 0.56

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 7/20 0.47
ALDH1A1 P00352 4/20 0.42
GAA P10253 2/20 0.42
KMT2A Q03164 1/20 0.42
MAPT P10636 4/20 0.41
PTGER4 P35408 5/20 0.41
KDM5A P29375 1/20 0.41
KDM4C Q9H3R0 1/20 0.41
KDM5B Q9UGL1 1/20 0.41
RAB9A P51151 2/20 0.40
RECQL P46063 1/20 0.40
POLB P06746 1/20 0.40
PKM P14618 1/20 0.40
NPC1 O15118 1/20 0.39
SMN1; SMN2 Q16637 1/20 0.39
NR1I2 O75469 1/20 0.38
LMNA P02545 1/20 0.38
AHR P35869 1/20 0.38
ADORA3 P0DMS8 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14487048 0.85 BRD4 (0.43) KDM4EKMT2AMAPTPTGER4KDM5A
SCHEMBL2723759 0.81 LCK (0.41) KDM4EKDM5AKDM4CKDM5BPOLB
SCHEMBL23367117 0.81 KDM5A (0.41) KDM4EMAPTPTGER4KDM5AKDM4C
SCHEMBL31539885 0.80 CYP1A2 (0.41) ALDH1A1KMT2AMAPTPTGER4KDM5A
SCHEMBL17324739 0.80 KDM5A (0.42) KDM4EALDH1A1GAAKMT2AMAPT
SCHEMBL1563562 0.80 KDM5A (0.48) KDM4EALDH1A1MAPTPTGER4KDM5A
Hydrochloric Acid SCHEMBL23354423 0.79 KDM5A (0.40) KDM4EMAPTPTGER4KDM5AKDM4C
SCHEMBL1562180 0.79 ALDH1A1 (0.49) KDM4EALDH1A1KMT2AKDM5AKDM4C
SCHEMBL3589934 0.78 KDM5A (0.41) KDM4EMAPTPTGER4KDM5AKDM4C
Methane SCHEMBL27733031 0.78 KDM5A (0.47) KDM4EALDH1A1MAPTPTGER4KDM5A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-101466703-A Heterocyclic GABA-alpha subtype selective receptor modulators HOFFMANN LA ROCHE (CH) 2009-06-24 CN disclosed