SCHEMBL27745778

SCHEMBL27745778

Oc1ccc(Cl)c2cnc(N(c3ccccc3)N3CCOCC3)nc12

nearest known ligand 0.37

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 4/20 0.37
LMNA P02545 2/20 0.37
METAP2 P50579 2/20 0.37
MAPT P10636 2/20 0.37
BRD4 O60885 1/20 0.37
HSP90AA1 P07900 1/20 0.37
METAP1 P53582 1/20 0.37
PKM P14618 1/20 0.36
PIM1 P11309 1/20 0.35
KDM4A O75164 1/20 0.35
HPGD P15428 2/20 0.34
TSHR P16473 2/20 0.34
HSD17B10 Q99714 2/20 0.34
CNR2 P34972 1/20 0.33
ALDH1A1 P00352 2/20 0.33
GAA P10253 2/20 0.33
KMT2A Q03164 2/20 0.33
GLA P06280 1/20 0.33
NPC1 O15118 2/20 0.32
RAB9A P51151 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27745785 0.72 KDM4E (0.34) KDM4ELMNAMAPTMETAP1PKM
SCHEMBL18335244 0.72 METAP1 (0.43) KDM4ELMNAMAPTMETAP1PKM
SCHEMBL28865660 0.69 CDK2 (0.40) KDM4ELMNAPKMTSHRALDH1A1
SCHEMBL3131793 0.69 CHEK1 (0.35) KDM4ELMNAMAPTMETAP1PKM
SCHEMBL12614645 0.69 NPC1 (0.39) KDM4ELMNAPKMTSHRALDH1A1
SCHEMBL27794438 0.67 PIK3CA (0.39) KDM4ELMNAL3MBTL1PIK3CAMTOR
SCHEMBL27760171 0.67 KMT2A (0.44) LMNAMETAP2MAPTMETAP1ALDH1A1
SCHEMBL1633833 0.67 CDK2 (0.60) BRD4
SCHEMBL6100741 0.66 FGFR1 (0.40) KDM4ELMNAMAPTMETAP1PKM
SCHEMBL27801283 0.66 HTT (0.39) KDM4EMAPTALDH1A1KMT2AL3MBTL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-101454294-A Quinazolines for pdk1 inhibition NOVARTIS AG (CH) 2009-06-10 CN disclosed