SCHEMBL28865660

SCHEMBL28865660

c1ccc(N(c2ncc3[nH]cnc3n2)N2CCOCC2)cc1

nearest known ligand 0.40

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
CDK2 P24941 1/20 0.40
CHEK1 O14757 3/20 0.40
SRC P12931 1/20 0.40
PIK3CA P42336 7/20 0.39
PIK3CG P48736 7/20 0.39
MTOR P42345 6/20 0.39
STAT3 P40763 1/20 0.37
ALDH1A1 P00352 1/20 0.35
KDM4E B2RXH2 1/20 0.35
PAK1 Q13153 2/20 0.35
PDPK1 O15530 1/20 0.35
MAPK1 P28482 1/20 0.35
PKM P14618 1/20 0.35
LMNA P02545 1/20 0.34
TSHR P16473 1/20 0.34
SCD O00767 1/20 0.34
PDE10A Q9Y233 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3131793 0.81 CHEK1 (0.35) CHEK1SRCPIK3CAPIK3CGMTOR
SCHEMBL18335244 0.74 METAP1 (0.43) PIK3CAALDH1A1KDM4EMAPK1PKM
SCHEMBL12614645 0.71 NPC1 (0.39) ALDH1A1KDM4EPKMLMNATSHR
SCHEMBL27745778 0.69 KDM4E (0.37) PIK3CAPIK3CGMTORALDH1A1KDM4E
SCHEMBL3128313 0.68 KDM1A (0.33) ALDH1A1KDM4EMAPK1LMNATSHR
SCHEMBL27745785 0.68 KDM4E (0.34) PIK3CAPIK3CGMTORALDH1A1KDM4E
SCHEMBL27801283 0.68 HTT (0.39) ALDH1A1KDM4EMAPK1
SCHEMBL336706 0.68 PIK3CD (0.50) CHEK1SRCPIK3CAALDH1A1KDM4E
SCHEMBL9900897 0.67 PKM (0.36) ALDH1A1KDM4EMAPK1PKMLMNA
SCHEMBL27760171 0.64 KMT2A (0.44) ALDH1A1MAPK1LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-106432239-B Purine compound, composition and purposes 大连医科大学 2018-10-30 CN disclosed