SCHEMBL27747871

SCHEMBL27747871

NCc1ccc(Nc2c(F)cccc2Cl)c(CC(=O)Oc2ccc(C(N)=S)cc2)c1

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PTGS2 P35354 8/20 0.49
PTGS1 P23219 4/20 0.49
ABCB11 O95342 2/20 0.49
NR1I3 Q14994 2/20 0.49
PPARG P37231 1/20 0.49
CAMK2A Q9UQM7 1/20 0.39
TTR P02766 2/20 0.36
KMT2A Q03164 2/20 0.36
LMNA P02545 2/20 0.36
USP2 O75604 1/20 0.36
CYP2C9 P11712 1/20 0.36
TBXA2R P21731 1/20 0.36
MAPK1 P28482 1/20 0.36
TLR7 Q9NYK1 1/20 0.35
AKR1B10 O60218 1/20 0.34
UGT1A9 O60656 1/20 0.34
TRPA1 O75762 1/20 0.34
MT-CO2 P00403 1/20 0.34
ALB P02768 1/20 0.34
CXCL8 P10145 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2880887 0.89 PTGS2 (0.64) PTGS2PTGS1ABCB11NR1I3PPARG
SCHEMBL2886958 0.81 PTGS2 (0.66) PTGS2PTGS1ABCB11NR1I3PPARG
SCHEMBL15267399 0.81 PTGS2 (0.65) PTGS2PTGS1ABCB11NR1I3PPARG
SCHEMBL2889216 0.80 TTR (0.57) PTGS2PTGS1ABCB11NR1I3CAMK2A
SCHEMBL14307499 0.74 PTGS2 (0.63) PTGS2PTGS1ABCB11NR1I3PPARG
SCHEMBL13688513 0.72 PTGS2 (0.66) PTGS2PTGS1ABCB11NR1I3PPARG
SCHEMBL2888394 0.72 PTGS2 (0.60) PTGS2PTGS1ABCB11NR1I3PPARG
SCHEMBL21401012 0.72 TTR (0.57) PTGS2PTGS1ABCB11NR1I3CAMK2A
SCHEMBL15267404 0.71 PTGS2 (0.62) PTGS2PTGS1ABCB11NR1I3PPARG
SCHEMBL2881532 0.71 TTR (0.59) PTGS2PTGS1ABCB11NR1I3CAMK2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-101501018-A Hydrogen sulfide derivatives of non-steroidal anti-inflammatory drugs ANTIBE THERAPEUTICS INC (CA) 2009-08-05 CN disclosed
CN-101490029-A 4-hydroxythiobenzamide derivatives of drugs ANTIBE THERAPEUTICS INC (CA) 2009-07-22 CN disclosed