SCHEMBL27749290

SCHEMBL27749290

OCc1cn(-c2cc[c]cc2)cn1

nearest known ligand 0.47

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
PDE3B Q13370 1/20 0.47
PDE3A Q14432 1/20 0.47
CPB1 P15086 3/20 0.36
CPB2 Q96IY4 3/20 0.36
SCD O00767 1/20 0.35
PDE10A Q9Y233 1/20 0.33
L3MBTL1 Q9Y468 2/20 0.32
KDM4E B2RXH2 2/20 0.32
NOTUM Q6P988 4/20 0.32
CYP1A2 P05177 1/20 0.31
CYP3A4 P08684 1/20 0.31
CYP2D6 P10635 1/20 0.31
CYP19A1 P11511 1/20 0.31
CYP2C9 P11712 1/20 0.31
CYP2C19 P33261 1/20 0.31
GRM5 P41594 1/20 0.31
GRM1 Q13255 1/20 0.31
MAPT P10636 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27648842 0.82 CYP1A2 (0.37) PDE3BPDE3ACPB1CPB2CYP1A2
SCHEMBL4433834 0.81 CPB2 (0.50) PDE3BPDE3ACPB1CPB2PDE10A
SCHEMBL4432563 0.79 NOTUM (0.51) PDE3BPDE3ACPB1CPB2KDM4E
SCHEMBL3426575 0.79 PDE3B (0.50) PDE3BPDE3ACPB1CPB2SCD
SCHEMBL2173293 0.79 PDE3B (0.50) PDE3BPDE3ACPB1CPB2SCD
SCHEMBL4434213 0.79 NOTUM (0.51) PDE3BPDE3ACPB1CPB2KDM4E
SCHEMBL4428918 0.79 PDE3B (0.53) PDE3BPDE3ACPB1CPB2SCD
SCHEMBL4427934 0.76 PDE3B (0.54) PDE3BPDE3ACPB1CPB2PDE10A
SCHEMBL6785441 0.75 NOTUM (0.55) PDE3BPDE3ACPB1CPB2NOTUM
SCHEMBL4425521 0.75 P2RX7 (0.55) PDE3BPDE3ACPB1CPB2KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-101490036-B Factor xa inhibitors MILLENNIUM PHARM INC 2013-07-17 CN disclosed
CN-101490036-A Factor XA inhibitors MILLENNIUM PHARM INC (US) 2009-07-22 CN disclosed