SCHEMBL27749772

SCHEMBL27749772

O=C(CF)Nc1ccc(S(=O)(=O)Nc2nccs2)c2cccnc12

nearest known ligand 0.63

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 2/20 0.43
SCN3A Q9NY46 2/20 0.43
LMNA P02545 1/20 0.42
TSHR P16473 1/20 0.42
SMN1; SMN2 Q16637 1/20 0.42
ALDH1A1 P00352 1/20 0.42
PKM P14618 2/20 0.42
SLC40A1 Q9NP59 1/20 0.41
MEN1 O00255 1/20 0.41
KMT2A Q03164 1/20 0.41
RXFP1 Q9HBX9 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13007613 0.90 RXFP1 (0.45) SCN3ALMNATSHRSMN1; SMN2ALDH1A1
SCHEMBL8244471 0.87 KDM4E (0.47) KDM4ESCN3ALMNATSHRSMN1; SMN2
SCHEMBL1863465 0.86 SLC40A1 (0.51) KDM4EALDH1A1SLC40A1MEN1KMT2A
SCHEMBL8244222 0.85 NPC1 (0.57) SCN3ASMN1; SMN2ALDH1A1PKMMEN1
SCHEMBL1856352 0.82 KDM4E (0.53) KDM4ESMN1; SMN2ALDH1A1MEN1KMT2A
SCHEMBL1857366 0.81 SLC40A1 (0.45) SCN3ASMN1; SMN2ALDH1A1PKMSLC40A1
SCHEMBL11959664 0.80 POLB (0.47) KDM4ESMN1; SMN2ALDH1A1SLC40A1MEN1
SCHEMBL11959669 0.79 MAPK1 (0.48) KDM4ESCN3ALMNATSHRALDH1A1
SCHEMBL14962381 0.79 SLC40A1 (0.48) KDM4ESCN3ALMNAALDH1A1SLC40A1
SCHEMBL13007609 0.78 SCN3A (0.47) SCN3ASMN1; SMN2ALDH1A1PKMMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-101300253-B Bicyclic derivatives as modulators of voltage gated ion channels VERTEX PHARMA 2012-08-22 CN disclosed
CN-101300253-A Bicyclic derivatives as modulators of voltage gated ion channels VERTEX PHARMA (US) 2008-11-05 CN disclosed