SCHEMBL8244471

SCHEMBL8244471

O=C(O)Nc1ccc(S(=O)(=O)Nc2nccs2)c2cccnc12

nearest known ligand 0.70

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 2/20 0.47
ALDH1A1 P00352 2/20 0.45
MEN1 O00255 2/20 0.44
KMT2A Q03164 2/20 0.44
SCN3A Q9NY46 3/20 0.43
SCN1A P35498 1/20 0.43
SCN4A P35499 1/20 0.43
SCN5A Q14524 1/20 0.43
SCN9A Q15858 1/20 0.43
SCN2A Q99250 1/20 0.43
SCN8A Q9UQD0 1/20 0.43
SCN10A Q9Y5Y9 1/20 0.43
CYP3A4 P08684 1/20 0.43
PTGS1 P23219 1/20 0.43
MAPT P10636 2/20 0.43
USP2 O75604 1/20 0.43
ESR2 Q92731 1/20 0.43
HSD17B10 Q99714 1/20 0.43
LMNA P02545 1/20 0.43
TSHR P16473 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27749772 0.87 KDM4E (0.43) KDM4EALDH1A1MEN1KMT2ASCN3A
SCHEMBL1863465 0.87 SLC40A1 (0.51) KDM4EALDH1A1MEN1KMT2ASCN1A
SCHEMBL13007613 0.87 RXFP1 (0.45) ALDH1A1MEN1KMT2ASCN3ALMNA
SCHEMBL8244222 0.85 NPC1 (0.57) ALDH1A1MEN1KMT2ASCN3ASCN9A
SCHEMBL1856352 0.84 KDM4E (0.53) KDM4EALDH1A1MEN1KMT2ASCN1A
SCHEMBL1855121 0.83 KMT2A (0.63) MEN1KMT2ASCN3AHSD17B10LMNA
SCHEMBL11959669 0.82 MAPK1 (0.48) KDM4EALDH1A1MEN1KMT2ASCN3A
SCHEMBL11959664 0.82 POLB (0.47) KDM4EALDH1A1MEN1KMT2ASCN1A
SCHEMBL14962381 0.80 SLC40A1 (0.48) KDM4EALDH1A1MEN1KMT2ASCN3A
SCHEMBL1863212 0.80 KDM4E (0.51) KDM4EALDH1A1SCN9AMAPTUSP2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2007030618-A2 BICYCLIC DERIVATIVES AS MODULATORS OF VOLTAGE GATED ION CHANNELS VERTEX PHARMACEUTICALS INCORPORATED (US) 2007-03-15 WO disclosed