SCHEMBL27754643

SCHEMBL27754643

CC(C)(C)c1cc(C(C)(C)C)c([N+](=O)[O-])cc1O.CC(C)(C)c1cc([N+](=O)[O-])c(O)c(C(C)(C)C)c1

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GPR35 Q9HC97 4/20 0.51
SMN1; SMN2 Q16637 2/20 0.47
MEN1 O00255 2/20 0.47
KMT2A Q03164 2/20 0.47
HTT P42858 2/20 0.47
GALR3 O60755 1/20 0.47
L3MBTL1 Q9Y468 1/20 0.47
ALDH1A1 P00352 4/20 0.39
ALOX15 P16050 3/20 0.39
KDM4E B2RXH2 2/20 0.39
CYP1A2 P05177 2/20 0.39
MAPT P10636 2/20 0.39
ATP2A2 P16615 1/20 0.39
ATP2A3 Q93084 1/20 0.39
ALOX12 P18054 2/20 0.38
MAPK1 P28482 2/20 0.38
SNCA P37840 1/20 0.38
TTR P02766 1/20 0.38
CYP2C9 P11712 1/20 0.38
HPGD P15428 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL397532 0.89 GPR35 (0.62) GPR35SMN1; SMN2MEN1KMT2AHTT
SCHEMBL395354 0.86 ALDH1A1 (0.52) GPR35SMN1; SMN2MEN1KMT2AHTT
SCHEMBL31634157 0.80 ALDH1A1 (0.58) GPR35SMN1; SMN2MEN1KMT2AHTT
SCHEMBL690829 0.79 GPR35 (0.78) GPR35SMN1; SMN2MEN1KMT2AHTT
SCHEMBL1600577 0.79 GPR35 (0.57) GPR35SMN1; SMN2MEN1KMT2AHTT
SCHEMBL14210874 0.77 SMN1; SMN2 (0.46) GPR35SMN1; SMN2MEN1KMT2AHTT
SCHEMBL1600086 0.75 GPR35 (0.65) GPR35SMN1; SMN2MEN1KMT2AHTT
SCHEMBL769557 0.75 SMN1; SMN2 (0.44) GPR35SMN1; SMN2MEN1KMT2AHTT
SCHEMBL18467780 0.75 SMN1; SMN2 (0.44) GPR35SMN1; SMN2MEN1KMT2AHTT
SCHEMBL376977 0.75 SMN1; SMN2 (0.44) GPR35SMN1; SMN2MEN1KMT2AHTT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-101478964-B Compositions of N- [2, 4-bis (1, 1-dimethylethyl) -5-hydroxyphenyl ] -1, 4-dihydro-4-oxoquinoline-3-carboxamide VERTEX PHARMA CO LTD 2012-02-29 CN disclosed
CN-101478964-A Compositions of N- [2, 4-bis (1, 1-dimethylethyl) -5-hydroxyphenyl ] -1, 4-dihydro-4-oxoquinoline-3-carboxamide VERTEX PHARMA (US) 2009-07-08 CN disclosed
CN-101384172-A Solid forms of N- [2, 4-bis (1, 1-dimethylethyl) -5-hydroxyphenyl ] -1, 4-dihydro-4-oxoquinoline-3-carboxamide VERTEX PHARMA (US) 2009-03-11 CN disclosed