SCHEMBL27754653

SCHEMBL27754653

Nc1ccc(-c2ccccc2)c(NC(=O)c2cccc(-c3cccnc3)c2)c1

nearest known ligand 0.57

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HDAC1 Q13547 9/20 0.57
ABCB1 P08183 2/20 0.57
HDAC3 O15379 2/20 0.57
HDAC2 Q92769 2/20 0.57
KMO O15229 1/20 0.53
SIRT2 Q8IXJ6 2/20 0.50
ALDH1A1 P00352 1/20 0.49
TP53 P04637 1/20 0.49
MAPT P10636 1/20 0.49
GFER P55789 1/20 0.49
BLK P51451 1/20 0.48
BTK Q06187 1/20 0.48
MEN1 O00255 1/20 0.48
PSIP1 O75475 1/20 0.48
AXL P30530 1/20 0.48
MKNK1 Q9BUB5 1/20 0.48
MKNK2 Q9HBH9 1/20 0.48
SCN5A Q14524 2/20 0.48
SCN9A Q15858 2/20 0.48
ABL1 P00519 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27754689 0.90 HDAC1 (0.58) HDAC1ABCB1HDAC3HDAC2MKNK1
SCHEMBL4579819 0.81 HDAC1 (0.84) HDAC1ABCB1HDAC3HDAC2
SCHEMBL27775560 0.75 HDAC1 (0.58) HDAC1HDAC3HDAC2ALDH1A1MAPT
SCHEMBL7587070 0.75 HDAC1 (0.65) HDAC1ABCB1HDAC3HDAC2ALDH1A1
SCHEMBL1399704 0.75 KMO (0.67) HDAC1ABCB1HDAC3HDAC2KMO
SCHEMBL28125557 0.74 ALDH1A1 (0.54) HDAC1HDAC3HDAC2ALDH1A1TP53
SCHEMBL4578711 0.74 HDAC1 (0.84) HDAC1ABCB1HDAC3HDAC2
SCHEMBL27754673 0.73 HDAC1 (0.52) HDAC1HDAC3HDAC2MAPT
SCHEMBL28096618 0.73 KMO (0.69) ABCB1KMOSIRT2ALDH1A1MAPT
SCHEMBL13188259 0.73 KMO (0.69) HDAC1ABCB1HDAC3HDAC2KMO

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-101466670-B Inhibitors of histone deacetylase METHYLGENE INC 2013-04-17 CN claimed
CN-101466670-B Inhibitors of histone deacetylase METHYLGENE INC 2013-04-17 CN disclosed
CN-101466670-A Benzamide derivatives as inhibitors of histone deacetylase METHYLGENE INC (CA) 2009-06-24 CN disclosed