SCHEMBL2775558

SCHEMBL2775558

Cn1cc2c(C3CC3CNC(=O)O)cccc2n1

nearest known ligand 0.46

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
MTNR1B P49286 19/20 0.46
MTNR1A P48039 18/20 0.46
SLC6A4 P31645 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2776538 1.00 MTNR1B (0.46) MTNR1BMTNR1ASLC6A4
SCHEMBL2777449 1.00 MTNR1B (0.46) MTNR1BMTNR1ASLC6A4
SCHEMBL543708 0.91 MTNR1B (0.50) MTNR1BMTNR1ASLC6A4
SCHEMBL543564 0.91 MTNR1B (0.50) MTNR1BMTNR1ASLC6A4
SCHEMBL544113 0.91 MTNR1B (0.50) MTNR1BMTNR1ASLC6A4
SCHEMBL543467 0.89 MTNR1B (0.59) MTNR1BMTNR1ASLC6A4
SCHEMBL543804 0.89 MTNR1B (0.59) MTNR1BMTNR1ASLC6A4
SCHEMBL543691 0.89 MTNR1B (0.59) MTNR1BMTNR1ASLC6A4
SCHEMBL543466 0.89 MTNR1B (0.59) MTNR1BMTNR1ASLC6A4
SCHEMBL10257834 0.85 ADORA3 (0.42) MTNR1BMTNR1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2141150-B1 BICYCLIC COMPOUND AND PHARMACEUTICAL USE THEREOF TAKEDA PHARMACEUTICAL (JP) 2013-12-11 EP disclosed
EP-2141150-A1 BICYCLIC COMPOUND AND PHARMACEUTICAL USE THEREOF Takeda Pharmaceutical Company Limited (JP) 2010-01-06 EP disclosed