SCHEMBL2775562

SCHEMBL2775562

COCc1cc(C(=O)OC(=O)c2ccc(-c3ccccc3C)c(S(C)(=O)=O)c2)ccc1Br

nearest known ligand 0.36

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
S1PR1 P21453 6/20 0.36
S1PR3 Q99500 2/20 0.36
MAPT P10636 5/20 0.35
NPC1 O15118 4/20 0.35
RAB9A P51151 4/20 0.35
PTGS2 P35354 1/20 0.34
HTT P42858 2/20 0.34
POLB P06746 1/20 0.34
THRB P10828 1/20 0.34
PTGDR2 Q9Y5Y4 1/20 0.33
CNR1 P21554 1/20 0.33
CMA1 P23946 1/20 0.33
LMNA P02545 2/20 0.32
SMN1; SMN2 Q16637 2/20 0.32
ALDH1A1 P00352 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2775559 0.91 S1PR1 (0.41) S1PR1S1PR3MAPTHTTPOLB
SCHEMBL2771877 0.79 PTGS2 (0.52) MAPTNPC1RAB9APTGS2HTT
SCHEMBL2773164 0.74 PTGS2 (0.51) MAPTRAB9APTGS2POLBCMA1
SCHEMBL2772724 0.74 PTGS2 (0.41) MAPTPTGS2POLBPTGDR2SMN1; SMN2
SCHEMBL319975 0.74 S1PR1 (0.46) S1PR1S1PR3MAPTNPC1RAB9A
SCHEMBL2776075 0.72 TTR (0.50) MAPTPOLBSMN1; SMN2ALDH1A1
SCHEMBL256771 0.70 NOTUM (0.50) MAPTHTTPTGDR2LMNASMN1; SMN2
SCHEMBL30622268 0.70 NOTUM (0.50) MAPTHTTPTGDR2LMNASMN1; SMN2
SCHEMBL319590 0.70 S1PR1 (0.52) S1PR1S1PR3POLB
SCHEMBL3183891 0.70 CA12 (0.51) MAPTNPC1RAB9AHTTLMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2193125-A2 OXADIAZOLE DERIVATIVES Merck Serono S.A. (CH) 2010-06-09 EP disclosed
WO-2009043889-A2 OXADIAZOLE DERIVATIVES MERCK SERONO S.A. (CH) 2009-04-09 WO disclosed