SCHEMBL2773164

SCHEMBL2773164

COC(=O)c1ccc(-c2ccccc2C)c(S(C)(=O)=O)c1.Cc1ccccc1-c1ccc(C(=O)O)cc1S(C)(=O)=O

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PTGS2 P35354 1/20 0.51
RAD52 P43351 1/20 0.46
VCAM1 P19320 1/20 0.45
CMA1 P23946 1/20 0.44
KDM4E B2RXH2 2/20 0.44
PKM P14618 2/20 0.44
ALDH1A1 P00352 1/20 0.44
GAA P10253 1/20 0.44
HPGD P15428 1/20 0.44
TDP1 Q9NUW8 2/20 0.44
TTR P02766 1/20 0.42
PTPRC P08575 2/20 0.41
EGFR P00533 1/20 0.41
KDM6B O15054 1/20 0.41
KDM5C P41229 1/20 0.41
KDM4C Q9H3R0 1/20 0.41
KDM2A Q9Y2K7 1/20 0.41
KDM3A Q9Y4C1 1/20 0.41
PDK2 Q15119 1/20 0.41
TSHR P16473 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2771877 0.95 PTGS2 (0.52) PTGS2VCAM1CMA1KDM4EPKM
SCHEMBL2776075 0.91 TTR (0.50) RAD52KDM4EALDH1A1TDP1TTR
SCHEMBL2775559 0.80 S1PR1 (0.41) RAD52PKMALDH1A1TDP1TTR
SCHEMBL410258 0.79 PDK2 (0.51) PTGS2KDM4EALDH1A1GAAHPGD
SCHEMBL28268790 0.78 KDM4E (0.54) KDM4EALDH1A1GAAHPGDTDP1
SCHEMBL8895570 0.77 PTGS2 (0.60) PTGS2VCAM1CMA1KDM4EPKM
SCHEMBL408614 0.77 XDH (0.59) PTGS2KDM4EALDH1A1GAAHPGD
SCHEMBL30031799 0.76 VCAM1 (0.57) PTGS2VCAM1CMA1KDM4EALDH1A1
SCHEMBL1495428 0.76 VCAM1 (0.57) PTGS2VCAM1CMA1KDM4EALDH1A1
SCHEMBL2774426 0.76 PTGS2 (0.46) PTGS2KDM4EPKMALDH1A1GAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2193125-A2 OXADIAZOLE DERIVATIVES Merck Serono S.A. (CH) 2010-06-09 EP disclosed
WO-2009043889-A2 OXADIAZOLE DERIVATIVES MERCK SERONO S.A. (CH) 2009-04-09 WO disclosed