SCHEMBL27757809

SCHEMBL27757809

CC(C)(C)C(=O)ON1CCC(Nc2ccc(Br)cc2)CC1

nearest known ligand 0.49

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.49
MAPT P10636 2/20 0.48
NPC1 O15118 1/20 0.48
MAPK1 P28482 1/20 0.48
HTT P42858 1/20 0.48
RAB9A P51151 1/20 0.48
L3MBTL1 Q9Y468 1/20 0.48
CCR5 P51681 1/20 0.44
FPR2 P25090 4/20 0.42
FPR3 P25089 3/20 0.42
MEN1 O00255 2/20 0.41
KMT2A Q03164 2/20 0.41
EPHX2 P34913 1/20 0.41
ROCK2 O75116 2/20 0.39
CYP3A4 P08684 2/20 0.39
POLB P06746 1/20 0.39
PAK1 Q13153 1/20 0.39
CHRNA7 P36544 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27981483 0.88 ALDH1A1 (0.52) ALDH1A1MAPTNPC1MAPK1HTT
SCHEMBL27826414 0.86 ALDH1A1 (0.49) ALDH1A1MAPTNPC1MAPK1HTT
SCHEMBL27613627 0.86 ALDH1A1 (0.48) ALDH1A1MAPTNPC1MAPK1HTT
SCHEMBL27552067 0.84 ALDH1A1 (0.46) ALDH1A1MAPTNPC1MAPK1HTT
SCHEMBL27746449 0.81 KMT2A (0.40) ALDH1A1MAPTNPC1MAPK1HTT
SCHEMBL27976449 0.81 FPR2 (0.43) ALDH1A1NPC1RAB9AFPR2FPR3
SCHEMBL2873727 0.80 ALDH1A1 (0.75) ALDH1A1MAPTNPC1MAPK1HTT
SCHEMBL27756075 0.79 CDK12 (0.43)
SCHEMBL27629058 0.79 NAMPT (0.41) ALDH1A1MAPTHTTL3MBTL1FPR2
SCHEMBL15544585 0.78 POLB (0.46) ALDH1A1MAPTNPC1MAPK1HTT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-101415674-A Pyrrolidine derivatives as ERK inhibitors SCHERING CORP (US) 2009-04-22 CN disclosed
CN-100469767-C Bipiperidine derivatives and their use as chemokine receptor inhibitors NOVARTIS AG (CH) 2009-03-18 CN disclosed
CN-1501915-A Bipiperidine derivatives and their use as chemokine receptor inhibitors ��˹��ŵ�� 2004-06-02 CN disclosed