SCHEMBL27760418

SCHEMBL27760418

NC(=O)Cn1cncc1C(=O)O

nearest known ligand 0.38

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 1/20 0.38
TDP1 Q9NUW8 1/20 0.38
TRPA1 O75762 2/20 0.35
CYP11B1 P15538 4/20 0.32
CYP11B2 P19099 4/20 0.32
RXFP1 Q9HBX9 1/20 0.31
TBXAS1 P24557 1/20 0.31
MAPT P10636 1/20 0.30
GPBAR1 Q8TDU6 1/20 0.30
CYP1A2 P05177 2/20 0.30
CYP3A4 P08684 2/20 0.30
GABRA1 P14867 2/20 0.30
GABRB2 P47870 2/20 0.30
LMNA P02545 1/20 0.30
CYP2C9 P11712 1/20 0.30
CYP2C19 P33261 1/20 0.30
ABCB11 O95342 1/20 0.30
GABRA2 P47869 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9819383 0.77 ALDH1A1 (0.44) ALDH1A1TDP1CYP11B1CYP11B2CYP1A2
SCHEMBL1178676 0.76 CYP19A1 (0.39) TRPA1CYP11B1CYP11B2
SCHEMBL12821930 0.73 ALDH1A1 (0.41) ALDH1A1TDP1CYP11B1CYP11B2CYP1A2
SCHEMBL15202232 0.73 ALDH1A1 (0.37) ALDH1A1TDP1CYP11B1CYP11B2CYP1A2
SCHEMBL5487137 0.73 TRPA1 (0.40) ALDH1A1TDP1TRPA1RXFP1TBXAS1
SCHEMBL23354136 0.73 ALDH1A1 (0.37) ALDH1A1TDP1CYP11B1CYP11B2CYP1A2
SCHEMBL21879876 0.73 ALDH1A1 (0.47) ALDH1A1TDP1CYP11B1CYP11B2CYP1A2
SCHEMBL1950890 0.73 CYP11B1 (0.57) ALDH1A1CYP11B1CYP11B2MAPTCYP3A4
SCHEMBL23930976 0.71 ALDH1A1 (0.40) ALDH1A1TDP1CYP11B1CYP11B2TBXAS1
SCHEMBL31518413 0.71 ALDH1A1 (0.40) ALDH1A1TDP1CYP11B1CYP11B2MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-101420942-B Small-molecule modulators of TRP-P8 activity DENDREON CORP 2014-03-12 CN disclosed
CN-101420942-A Small-molecule modulators of TRP-P8 activity DENDREON CORP (US) 2009-04-29 CN disclosed