SCHEMBL27760686

SCHEMBL27760686

Oc1ccc(N2C=CC=NC2)cc1

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ENPP2 Q13822 1/20 0.36
MKNK1 Q9BUB5 1/20 0.36
MKNK2 Q9HBH9 1/20 0.36
KMT2A Q03164 3/20 0.33
MEN1 O00255 2/20 0.33
GAA P10253 1/20 0.33
MAPT P10636 3/20 0.32
PKM P14618 2/20 0.31
HSP90AA1 P07900 1/20 0.31
MAPK1 P28482 1/20 0.31
NPSR1 Q6W5P4 1/20 0.31
MGLL Q99685 1/20 0.31
TDP1 Q9NUW8 1/20 0.31
KDM4E B2RXH2 2/20 0.31
ALDH1A1 P00352 2/20 0.31
NPC1 O15118 1/20 0.31
CA12 O43570 1/20 0.31
GMNN O75496 1/20 0.31
CA1 P00915 1/20 0.31
CA2 P00918 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28261507 0.81 MAPK1 (0.33) KMT2AMEN1MAPTMAPK1MGLL
SCHEMBL28165369 0.80 CHKA (0.39) MAPTNPSR1TDP1LMNA
SCHEMBL2362320 0.80 MAPT (0.35) KMT2AMEN1GAAMAPTMAPK1
SCHEMBL27457816 0.79 MEN1 (0.41) KMT2AMEN1KDM4EALDH1A1NPC1
SCHEMBL27914491 0.78 TSHR (0.40) KMT2AMEN1MAPK1MGLLALDH1A1
SCHEMBL2115712 0.77
SCHEMBL27974239 0.77
SCHEMBL28249904 0.77 KIF11 (0.37) MAPTTDP1CA12CA2CYP3A4
SCHEMBL4576927 0.74
SCHEMBL27039521 0.74 ADRB2 (0.51) KDM4EALDH1A1LMNAHSD17B10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-101486711-B 2,3-diaryl pyrimidine [1,2-a]benzimidazole heterocyclic compound, preparation and use thereof UNIV SHANXI NORMAL 2011-07-06 CN disclosed
CN-101506175-A 2-anilino-4-(heterocyclic)amino-pyrimidines as inhibitors of protein kinase C-alpha BOEHRINGER INGELHEIM INT (DE) 2009-08-12 CN disclosed
CN-101486711-A 2,3-diaryl pyrimidine [1,2-a]benzimidazole heterocyclic compound, preparation and use thereof UNIV SHANXI NORMAL (CN) 2009-07-22 CN disclosed