SCHEMBL27763045

SCHEMBL27763045

O=C(C=C(Cl)c1ccccc1)N1CCNCC1

nearest known ligand 0.58

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
SIGMAR1 Q99720 1/20 0.58
POLB P06746 1/20 0.45
USP2 O75604 1/20 0.45
ALDH1A1 P00352 1/20 0.45
TSHR P16473 1/20 0.45
HSD17B10 Q99714 1/20 0.45
RXFP1 Q9HBX9 1/20 0.45
ABCC1 P33527 1/20 0.40
MEN1 O00255 1/20 0.40
KMT2A Q03164 1/20 0.40
CCNC P24863 2/20 0.39
CDK8 P49336 2/20 0.39
OPRD1 P41143 1/20 0.39
GPR183 P32249 1/20 0.39
HRH4 Q9H3N8 1/20 0.38
HRH3 Q9Y5N1 1/20 0.38
HTR6 P50406 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27784855 0.81 SIGMAR1 (0.58) SIGMAR1POLBUSP2ALDH1A1TSHR
SCHEMBL27763340 0.79 SIGMAR1 (0.55) SIGMAR1POLBUSP2ALDH1A1TSHR
SCHEMBL27784857 0.77 SIGMAR1 (0.53) SIGMAR1POLBUSP2ALDH1A1TSHR
SCHEMBL27318407 0.76 SIGMAR1 (0.60) SIGMAR1POLBUSP2ALDH1A1TSHR
Benzamide SCHEMBL1474746 0.75 SIGMAR1 (0.58) SIGMAR1POLBUSP2ALDH1A1TSHR
SCHEMBL8937583 0.75 SIGMAR1 (0.49) SIGMAR1ALDH1A1RXFP1HRH4HTR6
SCHEMBL28393 0.74 SIGMAR1 (1.00) SIGMAR1POLBUSP2ALDH1A1TSHR
SCHEMBL894920 0.74 SIGMAR1 (1.00) SIGMAR1POLBUSP2ALDH1A1TSHR
SCHEMBL13899801 0.74 SIGMAR1 (0.62) SIGMAR1POLBUSP2ALDH1A1TSHR
SCHEMBL3999141 0.74 SIGMAR1 (0.62) SIGMAR1POLBUSP2ALDH1A1TSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-101591311-A 1-(3-phenyl acryloyl) bridged piperazine derivatives and preparation method thereof UNIV HEBEI TECHNOLOGY (CN) 2009-12-02 CN claimed
CN-101591311-A 1-(3-phenyl acryloyl) bridged piperazine derivatives and preparation method thereof UNIV HEBEI TECHNOLOGY (CN) 2009-12-02 CN disclosed