SCHEMBL27765697

SCHEMBL27765697

COc1cc(F)c(Br)c(F)c1C

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TUBB1 Q9H4B7 5/20 0.36
MAPT P10636 1/20 0.35
NPSR1 Q6W5P4 1/20 0.35
AKR1B1 P15121 1/20 0.35
PDE3B Q13370 2/20 0.33
PDE3A Q14432 2/20 0.33
POLB P06746 1/20 0.33
L3MBTL1 Q9Y468 1/20 0.33
ALDH1A1 P00352 1/20 0.33
TSHR P16473 1/20 0.33
PPARG P37231 1/20 0.33
NCOA2 Q15596 1/20 0.33
NCOA1 Q15788 1/20 0.33
SMN1; SMN2 Q16637 1/20 0.33
RXFP1 Q9HBX9 1/20 0.33
NQO2 P16083 1/20 0.33
ACHE P22303 2/20 0.32
CYP3A4 P08684 1/20 0.32
LMNA P02545 1/20 0.32
MAPK1 P28482 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20698169 0.83 TUBB1 (0.36) TUBB1MAPTNPSR1AKR1B1PDE3B
SCHEMBL6070092 0.83 MAPT (0.38) TUBB1MAPTNPSR1AKR1B1POLB
SCHEMBL27598496 0.82 ACHE (0.40) TUBB1MAPTNPSR1AKR1B1ALDH1A1
SCHEMBL8885005 0.80 TUBB1 (0.41) TUBB1MAPTL3MBTL1ALDH1A1RXFP1
SCHEMBL26607051 0.80 NPSR1 (0.36) MAPTNPSR1PDE3BPDE3APOLB
SCHEMBL27765600 0.77 ALDH1A1 (0.38) TUBB1MAPTNPSR1POLBL3MBTL1
SCHEMBL1491275 0.75 HDAC1 (0.35)
SCHEMBL9678363 0.74 TUBB1 (0.40) TUBB1MAPTNPSR1AKR1B1POLB
SCHEMBL6078582 0.73 NPSR1 (0.34) TUBB1MAPTNPSR1AKR1B1POLB
SCHEMBL6823575 0.73 ERN1 (0.47) TUBB1MAPTPOLBL3MBTL1ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-101421258-B Sulfonyl-substituted bicyclic compounds as PPAR modulators KALYPSYS INC 2013-08-21 CN disclosed
CN-101641335-A Amino-5-[substituted-4-(difluoromethoxy)phenyl]-5- phenylimidazolone compounds as ss-secretase inhibitors WYETH CORP US 2010-02-03 CN disclosed
CN-101421258-A Sulfonyl-substituted bicyclic compounds as PPAR modulators KALYSPSYS INC (US) 2009-04-29 CN disclosed