SCHEMBL27766643

SCHEMBL27766643

COc1nc(C)cn1C(c1ccccc1)(c1ccccc1)c1ccccc1

nearest known ligand 0.35

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SMN1; SMN2 Q16637 2/20 0.33
MEN1 O00255 1/20 0.32
OPRM1 P35372 1/20 0.32
OPRD1 P41143 1/20 0.32
KMT2A Q03164 1/20 0.32
NPSR1 Q6W5P4 1/20 0.32
CYP11B1 P15538 1/20 0.32
CYP11B2 P19099 1/20 0.32
ACSS2 Q9NR19 2/20 0.32
OGG1 O15527 1/20 0.32
EDNRB P24530 3/20 0.31
EDNRA P25101 3/20 0.31
POLB P06746 2/20 0.31
NR1I2 O75469 1/20 0.31
KCNE1 P15382 1/20 0.31
KCNQ1 P51787 1/20 0.31
F2RL3 Q96RI0 1/20 0.31
NQO2 P16083 1/20 0.31
MAPK1 P28482 1/20 0.31
MC4R P32245 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4884756 0.79 CYP11B1 (0.35) NPSR1CYP11B1CYP11B2MAPK1HSD17B10
SCHEMBL1423935 0.76 CYP11B1 (0.33) NPSR1CYP11B1CYP11B2GRM5
SCHEMBL8548870 0.76 NPSR1 (0.33) NPSR1CYP11B1CYP11B2GRM5
SCHEMBL20843903 0.74
SCHEMBL5326782 0.72 BRD4 (0.32) MEN1KMT2ANPSR1CYP11B1CYP11B2
SCHEMBL5447440 0.72 CYP19A1 (0.36) SMN1; SMN2MEN1OPRM1OPRD1KMT2A
SCHEMBL9408078 0.67 ALDH1A1 (0.36) SMN1; SMN2MEN1OPRM1OPRD1KMT2A
SCHEMBL27761432 0.66 CYP11B1 (0.31) CYP11B1CYP11B2ACSS2POLBNQO2
SCHEMBL3500675 0.66 CYP11B1 (0.33) NPSR1CYP11B1CYP11B2
SCHEMBL6197960 0.64 KDM4E (0.45) SMN1; SMN2MEN1KMT2ANPSR1MAPK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-101568542-B 5,6,7,8-tetrahydro-imidazo[1,5-a]pyrazine derivatives ACTELION PHARMACEUTICALS LTD 2013-03-27 CN disclosed
CN-101568542-A 5,6,7,8-tetrahydro-imidazo[1,5-a]pyrazine derivatives ACTELION PHARMACEUTICALS LTD (CH) 2009-10-28 CN disclosed