SCHEMBL27767010

SCHEMBL27767010

O=C(O)Cc1cncn1C1CCc2cc(F)ccc21

nearest known ligand 0.41

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
CYP17A1 P05093 2/20 0.41
CYP11B2 P19099 3/20 0.39
NPY5R Q15761 3/20 0.39
CYP19A1 P11511 1/20 0.38
CYP11B1 P15538 1/20 0.38
HRH1 P35367 1/20 0.38
KCNH2 Q12809 1/20 0.38
MAPK1 P28482 1/20 0.38
KDM4C Q9H3R0 2/20 0.37
KDM4A O75164 1/20 0.37
IDO1 P14902 1/20 0.36
TRPV1 Q8NER1 2/20 0.36
GCGR P47871 1/20 0.36
KDM5A P29375 1/20 0.36
KDM5B Q9UGL1 1/20 0.36
SRD5A1 P18405 3/20 0.36
MTNR1B P49286 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27788556 0.86 KDM4C (0.39) CYP11B2KDM4CIDO1TRPV1GCGR
SCHEMBL27767008 0.76 CYP17A1 (0.40) CYP17A1CYP11B2CYP19A1CYP11B1HRH1
SCHEMBL2817696 0.76 CYP17A1 (0.40) CYP17A1CYP11B2NPY5RCYP19A1CYP11B1
SCHEMBL4077603 0.67 FFAR1 (0.60)
SCHEMBL27788561 0.65 IDO1 (0.36) CYP11B2KDM4CIDO1
SCHEMBL8865733 0.65 CYP11B1 (0.62) CYP11B2CYP11B1
SCHEMBL1337775 0.64 PIN1 (0.50) MAPK1KDM4CTRPV1KDM5AKDM5B
SCHEMBL1340548 0.64 PIN1 (0.50) MAPK1KDM4CTRPV1KDM5AKDM5B
SCHEMBL1340154 0.64 PIN1 (0.50) MAPK1KDM4CTRPV1KDM5AKDM5B
SCHEMBL27788555 0.63 SRD5A1 (0.37) CYP11B2CYP11B1KDM4CTRPV1KDM5A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-101605777-A Imidazoles as aldosterone synthase inhibitors NOVARTIS AG (CH) 2009-12-16 CN disclosed