SCHEMBL8865733

SCHEMBL8865733

O=C(O)Cc1cncn1Cc1ccc(F)cc1

nearest known ligand 0.62

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
CYP11B1 P15538 17/20 0.62
CYP11B2 P19099 17/20 0.62
PTGDR2 Q9Y5Y4 1/20 0.43
GPBAR1 Q8TDU6 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2789150 0.86 CYP11B1 (0.61) CYP11B1CYP11B2
Hydrochloric Acid SCHEMBL8763109 0.85 CYP11B1 (0.60) CYP11B1CYP11B2
SCHEMBL2786255 0.82 CYP11B1 (0.71) CYP11B1CYP11B2
SCHEMBL7804285 0.81 FNTA (0.50) CYP11B1CYP11B2PTGDR2
Bromide SCHEMBL7927507 0.81 CYP11B1 (0.69) CYP11B1CYP11B2
Hydrochloric Acid SCHEMBL8481395 0.81 CYP11B1 (0.69) CYP11B1CYP11B2
Hydrochloric Acid SCHEMBL7748921 0.80 FNTA (0.49) CYP11B1CYP11B2PTGDR2
Hydrochloric Acid SCHEMBL7842775 0.80 CYP11B1 (0.67) CYP11B1CYP11B2
SCHEMBL17544540 0.79 CYP11B1 (0.71) CYP11B1CYP11B2GPBAR1
SCHEMBL7169286 0.79 CYP11B1 (0.57) CYP11B1CYP11B2GPBAR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5652257-A ANTICARCINOGENIC MERCK & CO., INC. (US) 1997-07-29 US disclosed
WO-1996010034-A2 THIOL-FREE INHIBITORS OF FARNESYL-PROTEIN TRANSFERASE MERCK & CO., INC. (US) 1996-04-04 WO disclosed