SCHEMBL27768209

SCHEMBL27768209

Cc1nc2c(s1)CCN(C(=O)c1ccc(COC(=O)C3CC3)c(C)c1)c1ccccc1-2

nearest known ligand 0.42

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
PDCD1 Q15116 5/20 0.42
CD274 Q9NZQ7 5/20 0.42
AVPR2 P30518 12/20 0.41
AVPR1A P37288 1/20 0.36
ROCK2 O75116 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2131662 0.85 AVPR2 (0.49) PDCD1CD274AVPR2
SCHEMBL2129587 0.84 PDCD1 (0.47) PDCD1CD274AVPR2AVPR1A
SCHEMBL27789716 0.82 PDCD1 (0.44) PDCD1CD274AVPR2
SCHEMBL27789677 0.81 PDCD1 (0.38) PDCD1CD274AVPR2AVPR1A
SCHEMBL2705200 0.79 AVPR2 (0.43) PDCD1CD274AVPR2AVPR1AROCK2
SCHEMBL2129812 0.77 SLC22A12 (0.46) PDCD1CD274AVPR2AVPR1AROCK2
SCHEMBL1495958 0.77 ALDH1A1 (0.50) AVPR2AVPR1A
SCHEMBL8556725 0.75 AVPR2 (0.48) AVPR2AVPR1A
SCHEMBL27789681 0.73 PDCD1 (0.38) PDCD1CD274AVPR2
SCHEMBL2704715 0.73 AVPR2 (0.45) PDCD1CD274AVPR2AVPR1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-101563347-A Vasopressin V1a antagonists VANTIA LTD (GB) 2009-10-21 CN disclosed