SCHEMBL27768291

SCHEMBL27768291

COc1ccc(CCN2CCN(CCOc3ccccc3-n3ccnc3)CC2)cc1OC

nearest known ligand 0.59

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
ADRA1D P25100 2/20 0.59
ADRA1A P35348 2/20 0.59
ADRA1B P35368 2/20 0.59
SIGMAR1 Q99720 4/20 0.52
EBP Q15125 2/20 0.52
TMEM97 Q5BJF2 1/20 0.52
TP53 P04637 1/20 0.48
CYP1A2 P05177 1/20 0.48
CYP3A4 P08684 1/20 0.48
CYP2D6 P10635 1/20 0.48
CYP2C9 P11712 1/20 0.48
TSHR P16473 1/20 0.48
NFKB1 P19838 1/20 0.48
CYP2C19 P33261 1/20 0.48
MTOR P42345 1/20 0.48
RAB9A P51151 1/20 0.48
HIF1A Q16665 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1332712 0.83 CYP2D6 (0.59) ADRA1DADRA1AADRA1BSIGMAR1EBP
SCHEMBL1334263 0.83 SIGMAR1 (0.68) ADRA1DADRA1AADRA1BSIGMAR1EBP
SCHEMBL12126795 0.79 SIGMAR1 (0.62) ADRA1DADRA1AADRA1BSIGMAR1EBP
SCHEMBL7030738 0.78 SIGMAR1 (0.61) ADRA1DADRA1AADRA1BSIGMAR1EBP
SCHEMBL12165084 0.78 SIGMAR1 (0.61) ADRA1DADRA1AADRA1BSIGMAR1EBP
SCHEMBL1332065 0.78 SIGMAR1 (0.61) ADRA1DADRA1AADRA1BSIGMAR1EBP
Hydrochloric Acid SCHEMBL1332727 0.77 SIGMAR1 (0.60) ADRA1DADRA1AADRA1BSIGMAR1EBP
SCHEMBL1332200 0.76 SIGMAR1 (0.69) ADRA1DADRA1AADRA1BSIGMAR1EBP
Hydrochloric Acid SCHEMBL1332118 0.75 SIGMAR1 (0.67) ADRA1DADRA1AADRA1BSIGMAR1EBP
SCHEMBL1333821 0.75 SIGMAR1 (0.58) ADRA1DADRA1AADRA1BSIGMAR1EBP

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-101511187-B Piperidine and piperazine derivatives MS SCIENCE CORP 2012-07-04 CN disclosed
CN-101448503-B Piperidine and piperazine derivatives MS SCIENCE CORP 2011-04-13 CN disclosed
CN-101511187-A Piperidine and piperazine derivatives MS SCIENCE CORP (JP) 2009-08-19 CN disclosed
CN-101448503-A Piperidine and piperazine derivatives MS SCIENCE CORP (JP) 2009-06-03 CN disclosed