SCHEMBL27768559

SCHEMBL27768559

CN(C=O)c1nnc(Cc2ccoc2)c2cc(-c3ccc(Cl)cc3)sc12

nearest known ligand 0.35

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
MCHR1 Q99705 2/20 0.35
FLT1 P17948 1/20 0.35
KDR P35968 1/20 0.35
CHEK1 O14757 3/20 0.34
STK17B O94768 1/20 0.31
MAP3K8 P41279 1/20 0.31
ACHE P22303 1/20 0.30
KDM4E B2RXH2 1/20 0.30
LMNA P02545 1/20 0.30
RAB9A P51151 1/20 0.30
SMN1; SMN2 Q16637 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27768365 0.84 CHEK1 (0.35) MCHR1FLT1KDRCHEK1STK17B
SCHEMBL29012242 0.82 FLT1 (0.42) FLT1KDRCHEK1LMNA
SCHEMBL12922013 0.81 CHEK1 (0.39) MCHR1CHEK1STK17BMAP3K8ACHE
SCHEMBL8827320 0.80 CHEK1 (0.49) MCHR1CHEK1STK17BMAP3K8ACHE
SCHEMBL12922014 0.78 CHEK1 (0.40) MCHR1CHEK1STK17BMAP3K8ACHE
SCHEMBL12922040 0.76 MAPT (0.41) CHEK1STK17BACHE
SCHEMBL28776699 0.76 CHEK1 (0.34) CHEK1STK17BMAP3K8KDM4ELMNA
SCHEMBL28781348 0.75 MCHR1 (0.39) MCHR1CHEK1
SCHEMBL26983380 0.74 MCHR1 (0.35) MCHR1CHEK1
SCHEMBL27768315 0.73 CHEK1 (0.41) MCHR1CHEK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-115038439-A Combination cancer therapy with CHK inhibitors 上海华禹生物科技有限公司 2022-09-09 CN claimed
CN-115038440-A Combination cancer therapy with CHK inhibitors 上海华禹生物科技有限公司 2022-09-09 CN claimed
CN-101481380-A Thiofuran pyridazine compound, preparation thereof, pharmaceutical composition and uses thereof ZHEJIANG MEDICINE CO LTD (CN) 2009-07-15 CN claimed
CN-115038439-A Combination cancer therapy with CHK inhibitors 上海华禹生物科技有限公司 2022-09-09 CN disclosed
CN-115038440-A Combination cancer therapy with CHK inhibitors 上海华禹生物科技有限公司 2022-09-09 CN disclosed
CN-101481380-A Thiofuran pyridazine compound, preparation thereof, pharmaceutical composition and uses thereof ZHEJIANG MEDICINE CO LTD (CN) 2009-07-15 CN disclosed