SCHEMBL27768759

SCHEMBL27768759

c1ccc(CCNCc2ccc3ncc4cccn4c3c2)cc1

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GAA P10253 2/20 0.49
KDM4E B2RXH2 2/20 0.49
ALDH1A1 P00352 2/20 0.49
GLA P06280 1/20 0.49
HPGD P15428 1/20 0.49
HSD17B10 Q99714 1/20 0.49
MAPT P10636 1/20 0.43
CYP3A4 P08684 2/20 0.43
CYP2D6 P10635 2/20 0.43
CYP2C19 P33261 2/20 0.43
ROCK2 O75116 1/20 0.43
KCNH2 Q12809 1/20 0.43
ROCK1 Q13464 1/20 0.43
BCHE P06276 7/20 0.42
SLC2A1 P11166 1/20 0.41
EPHX2 P34913 1/20 0.40
NLRP3 Q96P20 1/20 0.39
HDAC1 Q13547 1/20 0.38
CA12 O43570 1/20 0.38
CA1 P00915 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27768407 0.90 KDM4E (0.54) GAAKDM4EALDH1A1GLAHPGD
SCHEMBL27768416 0.80 KDM4E (0.54) GAAKDM4EALDH1A1GLAHPGD
SCHEMBL27768388 0.77 KDM4E (0.44) GAAKDM4EALDH1A1GLAHPGD
SCHEMBL27768414 0.77 PARP1 (0.51) GAAKDM4EALDH1A1GLAHPGD
SCHEMBL27789949 0.77 KDM4E (0.49) GAAKDM4EALDH1A1GLAHPGD
SCHEMBL27768404 0.75 ALDH1A1 (0.47) GAAKDM4EALDH1A1GLAHPGD
SCHEMBL27789942 0.74 ALDH1A1 (0.46) GAAKDM4EALDH1A1GLAHPGD
SCHEMBL27789947 0.73 KDM4E (0.45) GAAKDM4EALDH1A1GLAHPGD
SCHEMBL27768390 0.70 ALDH1A1 (0.50) GAAKDM4EALDH1A1GLAHPGD
SCHEMBL27768389 0.69 PARP1 (0.49) GAAKDM4EALDH1A1GLAHPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-101616919-B Poly (ADP ribose) polymerase inhibitors ABBOTT LAB 2012-10-10 CN claimed
CN-101616919-B Poly (ADP ribose) polymerase inhibitors ABBOTT LAB 2012-10-10 CN disclosed
CN-101616919-A Poly (ADP ribose) polymerase inhibitors ABBOTT LAB 2009-12-30 CN disclosed