SCHEMBL27769441

SCHEMBL27769441

Cc1ccc(C[CH]Cc2ccc(F)c(C)c2)cc1

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SIGMAR1 Q99720 2/20 0.39
DRD4 P21917 1/20 0.39
TMEM97 Q5BJF2 1/20 0.39
NFE2L2 Q16236 1/20 0.39
SLC6A2 P23975 1/20 0.39
SLC6A4 P31645 1/20 0.39
SLC6A3 Q01959 1/20 0.39
DAO P14920 1/20 0.39
MMP13 P45452 1/20 0.37
CYP1A2 P05177 1/20 0.36
CYP2A6 P11509 1/20 0.36
TAAR1 Q96RJ0 1/20 0.36
HDAC3 O15379 1/20 0.35
HDAC1 Q13547 1/20 0.35
HDAC2 Q92769 1/20 0.35
HDAC8 Q9BY41 1/20 0.35
IDO1 P14902 1/20 0.34
MPO P05164 1/20 0.34
ACHE P22303 2/20 0.33
DHODH Q02127 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27790908 0.87 SLC6A4 (0.38) SIGMAR1DRD4TMEM97SLC6A2SLC6A4
SCHEMBL9064997 0.79 IDO1 (0.50) CYP1A2CYP2A6TAAR1IDO1ACHE
SCHEMBL22148972 0.79 ESR1 (0.47) SIGMAR1DRD4TMEM97NFE2L2SLC6A2
SCHEMBL2370050 0.79 DAO (0.45) SLC6A2SLC6A4SLC6A3DAOMMP13
SCHEMBL7687745 0.79 SLC6A2 (0.41) SIGMAR1DRD4TMEM97SLC6A2SLC6A4
SCHEMBL27769496 0.78 MMP13 (0.39) SLC6A2SLC6A4SLC6A3DAOMMP13
SCHEMBL27769498 0.76 MMP13 (0.35) SLC6A2SLC6A4SLC6A3DAOMMP13
SCHEMBL27790940 0.75 MMP13 (0.36) SLC6A2SLC6A4SLC6A3DAOMMP13
SCHEMBL2090687 0.74 SLC6A2 (0.47) SIGMAR1DRD4TMEM97SLC6A2SLC6A4
SCHEMBL27769481 0.74 PPARD (0.39) DAOMMP13PTGS1PTGS2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-101627007-A Aminoamides as orexin antagonists HOFFMANN LA ROCHE 2010-01-13 CN claimed
CN-101627007-A Aminoamides as orexin antagonists HOFFMANN LA ROCHE 2010-01-13 CN disclosed