SCHEMBL27769481

SCHEMBL27769481

Cc1cc(C[CH]Cc2ccc(C(F)(F)F)nc2)ccc1F

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PPARD Q03181 1/20 0.39
DAO P14920 3/20 0.38
CYP2C9 P11712 2/20 0.37
TKT P29401 1/20 0.37
TRPV4 Q9HBA0 1/20 0.37
MMP13 P45452 1/20 0.36
KCNQ3 O43525 1/20 0.34
KCNQ2 O43526 1/20 0.34
KCNQ4 P56696 1/20 0.34
KCNQ5 Q9NR82 1/20 0.34
CYP2C19 P33261 1/20 0.34
GRIN1 Q05586 1/20 0.34
GRIN2B Q13224 1/20 0.34
NR1H2 P55055 1/20 0.34
NR1H3 Q13133 1/20 0.34
KDM1A O60341 1/20 0.34
MAOA P21397 1/20 0.34
MAOB P27338 1/20 0.34
PTGS1 P23219 1/20 0.34
PTGS2 P35354 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27769442 0.83 CYP2C9 (0.39) PPARDDAOCYP2C9TKTTRPV4
SCHEMBL27769496 0.82 MMP13 (0.39) DAOMMP13KCNQ3KCNQ2GRIN1
SCHEMBL27769444 0.77 ALDH1A1 (0.48) PPARDCYP2C9CYP2C19CYP3A4
SCHEMBL27791003 0.75 LOXL2 (0.41) DAOCYP2C9TRPV4KDM1AMAOA
SCHEMBL27769441 0.74 SIGMAR1 (0.39) DAOMMP13PTGS1PTGS2
SCHEMBL27790940 0.73 MMP13 (0.36) DAOMMP13GRIN1GRIN2BCYP3A4
SCHEMBL27769529 0.73 TKT (0.40) PPARDDAOTKTTRPV4KCNQ3
SCHEMBL27790908 0.72 SLC6A4 (0.38) DAOMMP13MAOAMAOB
SCHEMBL27790928 0.72 TKT (0.37) PPARDDAOTKTTRPV4KCNQ3
SCHEMBL3743226 0.72 PIM1 (0.42) PPARDDAOTKTMMP13KCNQ3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-101627007-A Aminoamides as orexin antagonists HOFFMANN LA ROCHE 2010-01-13 CN claimed
CN-101627007-A Aminoamides as orexin antagonists HOFFMANN LA ROCHE 2010-01-13 CN disclosed