SCHEMBL27773730

SCHEMBL27773730

C[CH]c1c[nH]c2cnccc12

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
DYRK1A Q13627 11/20 0.51
NFATC1 O95644 6/20 0.51
GSK3B P49841 4/20 0.51
CDK2 P24941 2/20 0.45
DYRK1B Q9Y463 2/20 0.45
PDPK1 O15530 1/20 0.45
TGFBR1 P36897 1/20 0.45
IKBKE Q14164 1/20 0.45
CCNT1 O60563 2/20 0.43
CDK9 P50750 2/20 0.43
HASPIN Q8TF76 2/20 0.43
IGF1R P08069 1/20 0.43
HTR2A P28223 1/20 0.41
KDM4E B2RXH2 1/20 0.39
GABRP O00591 1/20 0.39
GABRD O14764 1/20 0.39
IKBKB O14920 1/20 0.39
AURKA O14965 1/20 0.39
CHUK O15111 1/20 0.39
ALDH1A1 P00352 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2268299 0.81 CCNT1 (0.62) DYRK1ANFATC1GSK3BCDK2DYRK1B
SCHEMBL29664462 0.81 CCNT1 (0.62) DYRK1ANFATC1GSK3BCDK2DYRK1B
Hydrochloric Acid SCHEMBL3831446 0.80 CCNT1 (0.60) DYRK1ANFATC1GSK3BCDK2DYRK1B
SCHEMBL4268142 0.77 CCNT1 (0.65) DYRK1ANFATC1GSK3BCDK2DYRK1B
SCHEMBL4268145 0.77 CCNT1 (0.65) DYRK1ANFATC1GSK3BCDK2DYRK1B
SCHEMBL2619228 0.75 DYRK1A (0.56) DYRK1ANFATC1GSK3BCDK2DYRK1B
SCHEMBL6753342 0.74 APP (0.63) DYRK1ANFATC1GSK3BPDPK1TGFBR1
SCHEMBL315329 0.72 CYP2A6 (0.64) KDM4EALDH1A1HPGDSMN1; SMN2
SCHEMBL18746021 0.71 DYRK1A (0.56) DYRK1ANFATC1GSK3BCDK2DYRK1B
SCHEMBL245511 0.71 DYRK1A (0.61) DYRK1ANFATC1GSK3BCDK2DYRK1B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-101646656-B Pyrimidine hydrazide compounds as PGDS inhibitors SANOFI AVENTIS SPA 2013-08-14 CN disclosed
CN-101646656-A Pyrimidine hydrazide compounds as the PGDS inhibitor SANOFI AVENTIS FR 2010-02-10 CN disclosed