SCHEMBL27773795

SCHEMBL27773795

O=C1Cc2c(ccc(F)c2-c2c(F)cccc2F)N1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TDP2 O95551 1/20 0.40
AHR P35869 3/20 0.39
PDK2 Q15119 1/20 0.39
DRD2 P14416 3/20 0.39
DRD4 P21917 2/20 0.39
DRD3 P35462 2/20 0.39
SRD5A1 P18405 1/20 0.39
PGR P06401 1/20 0.39
GRIA1 P42261 1/20 0.39
CACNG8 Q8WXS5 1/20 0.39
CMA1 P23946 1/20 0.39
LMNA P02545 2/20 0.38
KDM4E B2RXH2 1/20 0.38
CHRM2 P08172 1/20 0.38
CYP3A4 P08684 1/20 0.38
HTR1A P08908 1/20 0.38
ADRA2A P08913 1/20 0.38
CYP2D6 P10635 1/20 0.38
CYP2C9 P11712 1/20 0.38
ADRA2B P18089 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3139769 0.86 PGR (0.43) DRD2DRD4DRD3SRD5A1PGR
SCHEMBL29622013 0.82 AHR (0.48) AHRPDK2DRD2DRD4DRD3
SCHEMBL261277 0.82 AHR (0.48) AHRPDK2DRD2DRD4DRD3
SCHEMBL153534 0.81 CCNB2 (0.44) AHRPDK2DRD2DRD4DRD3
SCHEMBL2076100 0.78 AHR (0.43) AHRPDK2DRD2DRD4DRD3
SCHEMBL22904178 0.75 TDP2 (0.64) TDP2AHRPDK2SRD5A1MEN1
SCHEMBL23252642 0.75 AHR (0.41) AHRPDK2DRD2DRD4DRD3
SCHEMBL19235316 0.75 AHR (0.41) AHRPDK2DRD2DRD4DRD3
SCHEMBL3136744 0.75 AHR (0.41) TDP2AHRPDK2DRD2DRD4
SCHEMBL31414332 0.75 AHR (0.49) TDP2AHRPDK2DRD2DRD4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-101675061-A pyrrolo-N-heterocyclic derivatives, process for their preparation and their use in medicine SHANGHAI HENGRUI PHARM CO LTD 2010-03-17 CN disclosed