SCHEMBL27775464

SCHEMBL27775464

CCOC(=O)C(C)(C)c1cccc(CN)c1

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CNR2 P34972 7/20 0.45
LOXL2 Q9Y4K0 1/20 0.44
MAOB P27338 1/20 0.43
MMP8 P22894 1/20 0.43
PPARG P37231 1/20 0.42
PPARA Q07869 1/20 0.42
KDM4E B2RXH2 1/20 0.42
NPSR1 Q6W5P4 1/20 0.42
CYP1A2 P05177 1/20 0.41
CYP2C19 P33261 1/20 0.41
PIN1 Q13526 1/20 0.41
THRB P10828 1/20 0.41
ALDH1A1 P00352 1/20 0.40
RECQL P46063 1/20 0.40
F2 P00734 1/20 0.39
F10 P00742 1/20 0.39
PLG P00747 1/20 0.39
PRSS1 P07477 1/20 0.39
RORC P51449 1/20 0.39
ENPP2 Q13822 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13140894 0.87 CNR2 (0.46) CNR2MAOBMMP8PPARGPPARA
SCHEMBL12585628 0.86 PPARA (0.50) CNR2MAOBMMP8PPARGPPARA
SCHEMBL13141048 0.86 IDO1 (0.51) CNR2MAOBMMP8PPARGPPARA
SCHEMBL2060663 0.85 CNR2 (0.45) CNR2MAOBMMP8PPARGPPARA
SCHEMBL14232380 0.85 LOXL2 (0.54) CNR2LOXL2MAOBCYP1A2CYP2C19
SCHEMBL15630699 0.84 RORC (0.51) CNR2LOXL2MAOBMMP8PPARA
Hydrochloric Acid SCHEMBL15609606 0.83 RORC (0.50) CNR2LOXL2MAOBMMP8PPARA
SCHEMBL6580520 0.83 PPARA (0.46) CNR2MAOBMMP8PPARGPPARA
SCHEMBL6161136 0.82 CNR2 (0.50) CNR2MAOBMMP8KDM4ECYP1A2
SCHEMBL2060134 0.81 CNR2 (0.52) CNR2MAOBMMP8PPARGPPARA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-103003266-A Hydroxyalkylbenzylpyrazoles and their use for the treatment of hyperproliferative and angiogenic diseases BAYER IP GMBH 2013-03-27 CN disclosed
CN-101668747-B Tetrahydroisoquinolin-1-one derivatives or salts thereof ASTELLAS PHARMA INC. (JP) 2012-02-01 CN disclosed
CN-101668747-A Tetrahydroisoquinolin-1-one derivatives or salts thereof ASTELLAS PHARMA INC 2010-03-10 CN disclosed