SCHEMBL27780446

SCHEMBL27780446

Br[Mg]Br.[c]1cccc(CN2CCOCC2)c1

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NCF1 P14598 1/20 0.48
HRH3 Q9Y5N1 2/20 0.47
ALDH1A1 P00352 2/20 0.46
MEN1 O00255 1/20 0.46
KMT2A Q03164 1/20 0.46
HTT P42858 3/20 0.43
KDM4E B2RXH2 1/20 0.43
HPGD P15428 1/20 0.43
CYP2A13 Q16696 5/20 0.43
SMN1; SMN2 Q16637 2/20 0.42
TSHR P16473 2/20 0.42
CXCR4 P61073 1/20 0.41
NOS1 P29475 2/20 0.41
NOS3 P29474 1/20 0.40
NOS2 P35228 1/20 0.40
NPC1 O15118 1/20 0.40
TP53 P04637 1/20 0.40
MAPK1 P28482 1/20 0.40
RAB9A P51151 1/20 0.40
POLB P06746 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL62595 0.94 HRH3 (0.53) NCF1HRH3ALDH1A1MEN1KMT2A
SCHEMBL27729376 0.92 HRH3 (0.51) NCF1HRH3ALDH1A1MEN1KMT2A
SCHEMBL27724955 0.86 SMN1; SMN2 (0.46) NCF1HRH3ALDH1A1KDM4ESMN1; SMN2
SCHEMBL27801847 0.84 SMN1; SMN2 (0.49) NCF1HRH3ALDH1A1KDM4ESMN1; SMN2
SCHEMBL27829415 0.84 HRH3 (0.54) NCF1HRH3ALDH1A1HTTKDM4E
SCHEMBL27809061 0.81 NCF1 (0.58) NCF1HRH3ALDH1A1HTTKDM4E
SCHEMBL27778712 0.81 HRH3 (0.58) NCF1HRH3ALDH1A1MEN1KMT2A
SCHEMBL23113743 0.79 HRH3 (0.47) NCF1HRH3ALDH1A1KDM4ESMN1; SMN2
SCHEMBL845155 0.79 HRH3 (0.52) NCF1HRH3ALDH1A1KDM4ESMN1; SMN2
SCHEMBL3149449 0.78 NCF1 (0.55) NCF1HRH3ALDH1A1HTTKDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-101652383-B Hepatitis c virus inhibitors BRISTOL MYERS SQUIBB CO 2013-09-18 CN disclosed
CN-102245613-A Phenyl and heteroaryl substituted thieno[2, 3-d] pyrimidines and their use as adenosine A2a receptor antagonists JANSSEN PHARMACEUTICA NV 2011-11-16 CN disclosed
CN-101652383-A Hepatitis c virus inhibitors SQUIBB BRISTOL MYERS CO US 2010-02-17 CN disclosed