SCHEMBL27809061

SCHEMBL27809061

[c]1cccc(CCc2cccc(CN3CCOCC3)c2)c1

nearest known ligand 0.58

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NCF1 P14598 1/20 0.58
HTT P42858 2/20 0.50
KDM4E B2RXH2 1/20 0.50
ALDH1A1 P00352 1/20 0.50
HPGD P15428 1/20 0.50
NOS1 P29475 1/20 0.47
HRH3 Q9Y5N1 4/20 0.44
BRD4 O60885 1/20 0.44
NPC1 O15118 1/20 0.43
TP53 P04637 1/20 0.43
TSHR P16473 1/20 0.43
MAPK1 P28482 1/20 0.43
RAB9A P51151 1/20 0.43
SMN1; SMN2 Q16637 1/20 0.43
PSMB8 P28062 1/20 0.43
CXCR4 P61073 1/20 0.42
PARP1 P09874 1/20 0.41
PRMT6 Q96LA8 1/20 0.41
CYP2A13 Q16696 1/20 0.41
CA2 P00918 2/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27829415 0.89 HRH3 (0.54) NCF1HTTKDM4EALDH1A1HPGD
SCHEMBL62595 0.87 HRH3 (0.53) NCF1HTTKDM4EALDH1A1HPGD
SCHEMBL27729376 0.85 HRH3 (0.51) NCF1HTTKDM4EALDH1A1HPGD
SCHEMBL28790869 0.83 SIGMAR1 (0.51) HRH3BRD4CXCR4PRMT6SIGMAR1
SCHEMBL3149449 0.83 NCF1 (0.55) NCF1HTTKDM4EALDH1A1HPGD
SCHEMBL11196105 0.82 NCF1 (0.83) NCF1HTTKDM4EALDH1A1HPGD
SCHEMBL27780446 0.81 NCF1 (0.48) NCF1HTTKDM4EALDH1A1HPGD
SCHEMBL5395459 0.81 SIGMAR1 (0.53) ALDH1A1POLBSIGMAR1
SCHEMBL4331617 0.81 AGXT (0.55) PRMT6SIGMAR1
SCHEMBL13959223 0.79 NCF1 (0.69) NCF1HTTKDM4EALDH1A1HPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-102046601-A Benzene or thiophene derivative and use thereof as VAP-1 inhibitor R TECH UENO LTD 2011-05-04 CN disclosed