SCHEMBL27780451

SCHEMBL27780451

CN1CCN(C(C(=O)N2CCC[C@H]2c2ncc(-c3cnc([C@@H]4CCCN4C(=O)[C@@H](c4ccccc4)N4CCCC4)[nH]3)[nH]2)c2ccccc2)CC1

nearest known ligand 0.52

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
OPRM1 P35372 2/20 0.48
OPRD1 P41143 2/20 0.48
KCNH2 Q12809 2/20 0.47
CYP3A4 P08684 3/20 0.47
CYP2C9 P11712 3/20 0.47
NR1I2 O75469 1/20 0.47
ABCB11 O95342 1/20 0.47
OPRK1 P41145 1/20 0.47
PRCP P42785 9/20 0.45
HCRTR1 O43613 1/20 0.43
HCRTR2 O43614 1/20 0.43
CYP1A2 P05177 2/20 0.42
CYP2D6 P10635 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19548078 0.94 KCNH2 (0.54) OPRM1OPRD1KCNH2CYP3A4CYP2C9
SCHEMBL1746897 0.94 KCNH2 (0.54) OPRM1OPRD1KCNH2CYP3A4CYP2C9
SCHEMBL14553283 0.93 OPRM1 (0.49) OPRM1OPRD1KCNH2CYP3A4CYP2C9
SCHEMBL27758910 0.89 OPRM1 (0.47) OPRM1OPRD1KCNH2CYP3A4CYP2C9
SCHEMBL27758903 0.89 ALDH1A1 (0.47) OPRM1OPRD1KCNH2CYP3A4CYP2C9
SCHEMBL1745425 0.88 CYP3A4 (0.57) OPRM1OPRD1KCNH2CYP3A4CYP2C9
SCHEMBL9284875 0.88 KCNH2 (0.55) OPRM1OPRD1KCNH2CYP3A4CYP2C9
SCHEMBL1747173 0.87 CYP3A4 (0.56) OPRM1OPRD1KCNH2CYP3A4CYP2C9
SCHEMBL1747178 0.87 CYP3A4 (0.56) OPRM1OPRD1KCNH2CYP3A4CYP2C9
SCHEMBL27758921 0.86 KCNH2 (0.48) OPRM1OPRD1KCNH2CYP3A4CYP2C9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-101558059-B Hepatitis c virus inhibitors BRISTOL MYERS SQUIBB CO 2014-12-03 CN claimed
CN-101558059-A Hepatitis C virus inhibitors BRISTOL MYERS SQUIBB CO (US) 2009-10-14 CN claimed