SCHEMBL27780474

SCHEMBL27780474

CNC1=C(C#N)C(c2ccc3c(c2)c(C)nn3C(=O)OC(C)(C)C)C(C#N)=C(NC)N1NC

nearest known ligand 0.36

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
GABRA1 P14867 1/20 0.36
TMEM97 Q5BJF2 1/20 0.36
MAP2K4 P45985 1/20 0.35
KDM4E B2RXH2 1/20 0.32
ALDH1A1 P00352 1/20 0.32
MAPT P10636 1/20 0.32
HPGD P15428 1/20 0.32
CASP1 P29466 1/20 0.32
HSD17B10 Q99714 1/20 0.32
GPR119 Q8TDV5 1/20 0.31
NR1H2 P55055 1/20 0.31
MET P08581 1/20 0.30
RPS6KA3 P51812 1/20 0.30
NR3C2 P08235 1/20 0.30
IRAK4 Q9NWZ3 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4995273 0.85 MET (0.41) GABRA1TMEM97MAP2K4KDM4EALDH1A1
SCHEMBL4985352 0.85 GABRA1 (0.48) GABRA1TMEM97MAP2K4KDM4EALDH1A1
SCHEMBL9906866 0.77 GABRA1 (0.41) GABRA1TMEM97MAP2K4KDM4EALDH1A1
SCHEMBL9906883 0.77 MET (0.35) GABRA1TMEM97MAP2K4METNR3C2
SCHEMBL1415058 0.76 GABRA1 (0.47) GABRA1TMEM97MAP2K4KDM4EALDH1A1
SCHEMBL4781102 0.75 GABRA1 (0.41) GABRA1MAP2K4GPR119NR1H2IRAK4
SCHEMBL4441866 0.75 GABRA1 (0.50) GABRA1TMEM97MAP2K4KDM4EALDH1A1
SCHEMBL4432848 0.73 GABRA1 (0.48) GABRA1TMEM97MAP2K4KDM4EALDH1A1
SCHEMBL3517327 0.72 MAP2K4 (0.44) GABRA1MAP2K4NR1H2
SCHEMBL931118 0.72 ELANE (0.43) MAP2K4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-101558040-A Dihydropyridine derivatives useful as protein kinase inhibitors BAYER SCHERING PHARMA AG (DE) 2009-10-14 CN disclosed