SCHEMBL27786396

SCHEMBL27786396

CC(C)(C)OC(N)=O.CCCn1cc(C(=O)N2CCC(N3C(=O)Cc4ccccc43)CC2)c2ccc(Cl)cc21

nearest known ligand 0.43

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
HSD11B1 P28845 1/20 0.43
AVPR1A P37288 4/20 0.43
CNR1 P21554 1/20 0.41
KCNH2 Q12809 1/20 0.41
OPRM1 P35372 1/20 0.40
OPRK1 P41145 1/20 0.40
OPRL1 P41146 1/20 0.40
TPSAB1 Q15661 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27786394 0.88 HSD11B1 (0.42) HSD11B1AVPR1ACNR1KCNH2
SCHEMBL829077 0.86 AVPR1A (0.49) HSD11B1AVPR1ACNR1KCNH2OPRM1
SCHEMBL828756 0.86 AVPR1A (0.47) HSD11B1AVPR1ACNR1OPRM1OPRK1
SCHEMBL825148 0.84 AVPR1A (0.59) HSD11B1AVPR1ACNR1OPRM1OPRK1
SCHEMBL825327 0.83 AVPR1A (0.47) HSD11B1AVPR1ACNR1OPRM1OPRK1
Hydrochloric Acid SCHEMBL829428 0.83 AVPR1A (0.46) HSD11B1AVPR1ACNR1OPRM1OPRK1
SCHEMBL825277 0.82 OXTR (0.49) HSD11B1AVPR1A
SCHEMBL825146 0.81 OXTR (0.50) HSD11B1AVPR1ACNR1OPRM1OPRK1
SCHEMBL825145 0.81 AVPR1A (0.50) HSD11B1AVPR1ACNR1KCNH2
SCHEMBL825238 0.81 AVPR1A (0.59) HSD11B1AVPR1ACNR1KCNH2OPRM1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-101583609-A Indoles HOFFMANN LA ROCHE (CH) 2009-11-18 CN disclosed