SCHEMBL27787484

SCHEMBL27787484

CC(=O)Oc1ccc(NCc2cc(Br)ccc2O)cc1C(=O)O

nearest known ligand 0.56

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
EGFR P00533 11/20 0.56
NOX4 Q9NPH5 3/20 0.56
ALDH1A1 P00352 2/20 0.56
MAPT P10636 2/20 0.56
TDP1 Q9NUW8 2/20 0.56
RGS12 O14924 1/20 0.56
LCK P06239 1/20 0.56
CAMKK2 Q96RR4 1/20 0.56
KDM4C Q9H3R0 1/20 0.55
CA1 P00915 2/20 0.51
CA2 P00918 2/20 0.51
CA12 O43570 1/20 0.51
CA9 Q16790 1/20 0.51
KDM4E B2RXH2 1/20 0.49
MEN1 O00255 1/20 0.49
USP2 O75604 1/20 0.49
GAA P10253 1/20 0.49
THRB P10828 1/20 0.49
ALOX15 P16050 1/20 0.49
CASP1 P29466 1/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27809392 0.93 EGFR (0.51) EGFRNOX4ALDH1A1MAPTTDP1
SCHEMBL28798414 0.88 EGFR (0.54) EGFRNOX4ALDH1A1MAPTTDP1
SCHEMBL27858209 0.88 EGFR (0.54) EGFRNOX4ALDH1A1MAPTTDP1
Lysine SCHEMBL27787482 0.87 EGFR (0.43) EGFRNOX4ALDH1A1MAPTTDP1
SCHEMBL27787480 0.86 EGFR (0.74) EGFRNOX4ALDH1A1MAPTTDP1
SCHEMBL27770270 0.82 EGFR (0.60) EGFRNOX4ALDH1A1MAPTTDP1
Lysine SCHEMBL27787481 0.81 CA1 (0.41) EGFRNOX4ALDH1A1MAPTTDP1
SCHEMBL28787539 0.79 EGFR (0.51) EGFRNOX4ALDH1A1MAPTTDP1
SCHEMBL11241726 0.77 CA1 (0.65) EGFRNOX4ALDH1A1MAPTTDP1
SCHEMBL25027 0.76 CFD (0.73) ALDH1A1TDP1KDM4EMEN1USP2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-102516107-A N-benzylaniline derivatives and application thereof UNIV NANJING MEDICAL 2012-06-27 CN disclosed
CN-101792399-A Aminosalicylic acid derivative lysine complex salt, preparation method and application thereof UNIV NANJING MEDICAL 2010-08-04 CN disclosed