SCHEMBL2779

SCHEMBL2779

CCCCC(=O)N(Cc1ccc(-c2ccccc2C#N)cc1Br)[C@H](C(=O)OCc1ccccc1)C(C)C

nearest known ligand 0.42

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
AGTR1 P30556 8/20 0.42
LTB4R2 Q9NPC1 7/20 0.41
ABCB11 O95342 1/20 0.41
GP6 Q9HCN6 1/20 0.41
FFAR1 O14842 2/20 0.36
AKR1B1 P15121 1/20 0.36
CYP2C9 P11712 1/20 0.33
S1PR1 P21453 1/20 0.33
OXTR P30559 1/20 0.33
AVPR1A P37288 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7276200 0.89 AGTR1 (0.48) AGTR1LTB4R2ABCB11GP6CYP2C9
SCHEMBL2140 0.88 AGTR1 (0.54) AGTR1LTB4R2ABCB11GP6FFAR1
SCHEMBL29378073 0.88 AGTR1 (0.54) AGTR1LTB4R2ABCB11GP6FFAR1
SCHEMBL1809623 0.88 AGTR1 (0.54) AGTR1LTB4R2ABCB11GP6FFAR1
SCHEMBL2780 0.86 FFAR1 (0.35) AGTR1FFAR1AKR1B1CYP2C9S1PR1
SCHEMBL2400 0.82 AGTR1 (0.48) AGTR1LTB4R2ABCB11GP6
SCHEMBL1975 0.82 AGTR1 (0.48) AGTR1LTB4R2ABCB11GP6
SCHEMBL2441623 0.82 AGTR1 (0.47) AGTR1LTB4R2ABCB11GP6FFAR1
SCHEMBL8483566 0.81 FFAR1 (0.42) AGTR1LTB4R2ABCB11GP6FFAR1
SCHEMBL14032861 0.80 LTB4R2 (0.44) AGTR1LTB4R2ABCB11GP6FFAR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5965592-A HYPOTENSIVE AGENTS NOVARTIS CORPORATION (US) 1999-10-12 US disclosed
EP-0443983-B1 Acyl compounds CIBA GEIGY AG (CH) 1996-02-28 EP disclosed
US-5399578-A Hypotensive; valsartan; high blood pressure and cardiac insufficiency CIBA-GEIGY CORP (US) 1995-03-21 US disclosed
EP-0443983-A1 Acyl compounds CIBA-GEIGY AG (CH) 1991-08-28 EP disclosed