SCHEMBL27795239

SCHEMBL27795239

Cc1cc(Cl)ncc1-c1cc(C(=O)N(C)c2ccccc2CCCCC(=O)O)ccc1Cl

nearest known ligand 0.42

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
GPBAR1 Q8TDU6 13/20 0.42
PTGDR2 Q9Y5Y4 1/20 0.37
RXRA P19793 1/20 0.35
RXRB P28702 1/20 0.35
FFAR4 Q5NUL3 1/20 0.35
RORC P51449 1/20 0.34
PPARD Q03181 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3339922 0.97 GPBAR1 (0.43) GPBAR1PTGDR2RXRARXRBFFAR4
SCHEMBL30509082 0.97 GPBAR1 (0.43) GPBAR1PTGDR2RXRARXRBFFAR4
SCHEMBL3339754 0.88 GPBAR1 (0.41) GPBAR1PTGDR2RORC
SCHEMBL30509078 0.88 GPBAR1 (0.41) GPBAR1PTGDR2RORC
SCHEMBL16390861 0.87 GPBAR1 (0.41) GPBAR1RXRARXRBFFAR4RORC
SCHEMBL3339509 0.83 RXRA (0.43) GPBAR1PTGDR2RXRARXRBRORC
SCHEMBL16858742 0.83 RXRA (0.38) GPBAR1PTGDR2RXRARXRBFFAR4
SCHEMBL3335704 0.82 GPBAR1 (0.50) GPBAR1RORC
SCHEMBL11263458 0.81 GPBAR1 (0.45) GPBAR1PTGDR2
SCHEMBL3337439 0.81 GPBAR1 (0.44) GPBAR1PTGDR2RORC

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-101678007-B Gonadotropin-releasing hormone receptor antagonists and its pharmaceutical application NEUROCRINE BIOSCIENCES INC 2013-07-03 CN disclosed
CN-101678007-A gonadotropin-releasing hormone receptor antagonists and methods relating thereto NEUROCRINE BIOSCIENCES INC 2010-03-24 CN disclosed