SCHEMBL27795243

SCHEMBL27795243

O=C(O)CCCCc1ccccc1NC(=O)c1ccc(Cl)c(Br)c1

nearest known ligand 0.61

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
SLC16A3 O15427 8/20 0.61
HDAC1 Q13547 4/20 0.46
HDAC8 Q9BY41 4/20 0.46
HDAC6 Q9UBN7 4/20 0.46
SUCNR1 Q9BXA5 3/20 0.45
F11 P03951 1/20 0.45
NR1H4 Q96RI1 3/20 0.45
PPARG P37231 2/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16390905 0.97 SLC16A3 (0.59) SLC16A3HDAC1HDAC8HDAC6SUCNR1
SCHEMBL3336081 0.84 SLC16A3 (0.53) SLC16A3HDAC1HDAC8HDAC6NR1H4
SCHEMBL3337087 0.81 SLC16A3 (0.42) SLC16A3HDAC1HDAC8HDAC6
SCHEMBL2229279 0.79 SLC16A3 (0.54) SLC16A3HDAC1NR1H4PPARG
SCHEMBL31661766 0.79 SLC16A3 (0.54) SLC16A3HDAC1NR1H4PPARG
SCHEMBL31661740 0.79 LMNA (0.56) SLC16A3SUCNR1F11PPARG
SCHEMBL2061475 0.79 LMNA (0.56) SLC16A3SUCNR1F11PPARG
SCHEMBL3554633 0.76 SLC16A3 (1.00) SLC16A3
SCHEMBL31661816 0.74 SMN1; SMN2 (0.53) SLC16A3PPARG
SCHEMBL13349339 0.73 MAPT (0.59) HDAC1HDAC8HDAC6PPARG

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-101678007-B Gonadotropin-releasing hormone receptor antagonists and its pharmaceutical application NEUROCRINE BIOSCIENCES INC 2013-07-03 CN disclosed
CN-101678007-A gonadotropin-releasing hormone receptor antagonists and methods relating thereto NEUROCRINE BIOSCIENCES INC 2010-03-24 CN disclosed