SCHEMBL27797271

SCHEMBL27797271

CCOc1cccc(OCC)c1/C=C\c1cccc(CCCN)c1

nearest known ligand 0.38

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
CYP1A1 P04798 1/20 0.38
CYP1A2 P05177 1/20 0.38
CYP1B1 Q16678 1/20 0.38
KDM4E B2RXH2 2/20 0.38
LMNA P02545 1/20 0.38
ALDH1A1 P00352 2/20 0.37
SMN1; SMN2 Q16637 1/20 0.37
AKR1C3 P42330 1/20 0.37
TAAR1 Q96RJ0 2/20 0.36
HDAC4 P56524 3/20 0.36
MEF2D Q14814 3/20 0.36
CALM1 P0DP23 1/20 0.36
EP300 Q09472 1/20 0.35
HTR6 P50406 1/20 0.35
TUBB1 Q9H4B7 1/20 0.35
EGFR P00533 1/20 0.35
RELA Q04206 1/20 0.35
CYP4F2 P78329 1/20 0.34
CYP4A11 Q02928 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8799051 1.00 CYP1A1 (0.38) CYP1A1CYP1A2CYP1B1KDM4ELMNA
SCHEMBL27955312 0.93 NFE2L2 (0.40) CYP1A1CYP1A2CYP1B1KDM4ELMNA
SCHEMBL4170999 0.87 NFE2L2 (0.43) CYP1A1CYP1A2CYP1B1KDM4ELMNA
SCHEMBL4170993 0.87 NFE2L2 (0.43) CYP1A1CYP1A2CYP1B1KDM4ELMNA
SCHEMBL4183387 0.86 CYP1A1 (0.54) CYP1A1CYP1A2CYP1B1KDM4ETAAR1
SCHEMBL4183390 0.86 CYP1A1 (0.54) CYP1A1CYP1A2CYP1B1KDM4ETAAR1
Ammonia Solution, Strong SCHEMBL27776433 0.85 CYP1A1 (0.41) CYP1A1CYP1A2CYP1B1KDM4ELMNA
SCHEMBL27776420 0.84 CYP1A1 (0.40) CYP1A1CYP1A2CYP1B1KDM4ELMNA
SCHEMBL28782912 0.80 CYP1A1 (0.41) CYP1A1CYP1A2CYP1B1KDM4ELMNA
SCHEMBL4161352 0.79 TAAR1 (0.45) TAAR1HDAC4MEF2DHTR6CYP4F2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-101686665-B Styrenyl derivative compounds for treating ophthalmic diseases and disorders ACUCELA INC 2014-04-23 CN claimed
CN-101686665-A styrenyl derivative compounds for treating ophthalmic diseases and disorders ACUCELA INC 2010-03-31 CN claimed
CN-101686665-A styrenyl derivative compounds for treating ophthalmic diseases and disorders ACUCELA INC 2010-03-31 CN disclosed