SCHEMBL27800296

SCHEMBL27800296

Cc1ccc(C(C)C(=O)C(C)c2ccc(C)nc2Nc2ccccc2)c(Nc2ccccc2)n1

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPT P10636 2/20 0.45
TP53 P04637 1/20 0.45
SMN1; SMN2 Q16637 1/20 0.45
ALDH1A1 P00352 2/20 0.43
OGG1 O15527 1/20 0.42
KMT2A Q03164 3/20 0.42
RAB9A P51151 3/20 0.42
MEN1 O00255 2/20 0.42
NPC1 O15118 2/20 0.42
GBA1 P04062 1/20 0.42
HPGD P15428 1/20 0.41
RXRA P19793 1/20 0.40
NR4A2 P43354 1/20 0.40
RXFP1 Q9HBX9 1/20 0.40
GAA P10253 1/20 0.40
CYP1A2 P05177 2/20 0.39
MDM2 Q00987 1/20 0.39
KDM4E B2RXH2 1/20 0.39
EGFR P00533 1/20 0.39
ITK Q08881 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27800314 0.81 TRPV1 (0.46) MAPTTP53SMN1; SMN2RAB9ANPC1
SCHEMBL27800307 0.80 ABCG2 (0.49) MAPTSMN1; SMN2ALDH1A1KMT2ARAB9A
SCHEMBL27779942 0.78 RAB9A (0.35) MAPTTP53ALDH1A1RAB9ANPC1
SCHEMBL27800317 0.78 DHODH (0.56) MAPTSMN1; SMN2ALDH1A1KMT2ARAB9A
SCHEMBL8171612 0.75 DHODH (0.57) MAPTTP53SMN1; SMN2ALDH1A1KMT2A
SCHEMBL846982 0.74 MAPT (0.44) MAPTTP53SMN1; SMN2ALDH1A1KMT2A
SCHEMBL27917422 0.73 IRAK4 (0.38) ALDH1A1RAB9ANPC1CYP1A2CYP2D6
SCHEMBL10169191 0.73 MAPK8 (0.54) MAPTSMN1; SMN2KMT2ARAB9ANPC1
SCHEMBL3636515 0.72 KDM4E (0.41) MAPTSMN1; SMN2ALDH1A1RAB9ANPC1
SCHEMBL12715339 0.72 MAPT (0.54) MAPTTP53SMN1; SMN2ALDH1A1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-101679270-B Dihydroquinone and dihydronaphthyridine inhibitors of JNK HOFFMANN LA ROCHE 2013-05-01 CN disclosed
CN-101679270-A Dihydroquinone and dihydronaphthyridine inhibitors of JNK HOFFMANN LA ROCHE 2010-03-24 CN disclosed