SCHEMBL27802443

SCHEMBL27802443

CN1CCN(c2cccc(-c3cc(-c4ccc(N(C(N)=O)c5ccc(Cl)c(C(F)(F)F)c5)cc4)[nH]n3)c2)CC1

nearest known ligand 0.51

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
PRKD1 Q15139 12/20 0.51
RAF1 P04049 5/20 0.48
BRAF P15056 5/20 0.48
MELK Q14680 1/20 0.46
LMNA P02545 1/20 0.40
SMN1; SMN2 Q16637 1/20 0.40
FLT3 P36888 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27823075 0.92 MELK (0.52) PRKD1RAF1BRAFMELKLMNA
SCHEMBL5523848 0.83 RAF1 (0.52) RAF1BRAFLMNAFLT3
SCHEMBL1790198 0.83 RAF1 (0.69) PRKD1RAF1BRAFMELKFLT3
SCHEMBL5534704 0.74 MELK (0.47) PRKD1MELKFLT3
SCHEMBL1791767 0.74 RAF1 (0.63) PRKD1RAF1BRAFMELKLMNA
SCHEMBL1081001 0.72 PRKD1 (0.73) PRKD1MELKFLT3
SCHEMBL3842420 0.72 PRKD1 (0.43) PRKD1MELKSMN1; SMN2FLT3
SCHEMBL3850883 0.71 BRD4 (0.46) PRKD1MELKSMN1; SMN2FLT3
SCHEMBL3850586 0.70 RET (0.46) PRKD1MELKSMN1; SMN2FLT3
SCHEMBL15104126 0.70 PRKD1 (0.46) PRKD1MELK

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-101959516-A Combination therapy comprising quinoxaline PI3K alpha inhibitors for the treatment of cancer EXELIXIS INC 2011-01-26 CN disclosed