SCHEMBL27804115

SCHEMBL27804115

Cc1ccc(N)cc1Cn1cc(CN(C)C)nn1

nearest known ligand 0.42

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
CHRNE Q04844 1/20 0.42
HSP90AB1 P08238 6/20 0.41
MAPK1 P28482 1/20 0.39
KMT2A Q03164 1/20 0.39
HDAC1 Q13547 1/20 0.37
NOTUM Q6P988 1/20 0.37
AMY1A P0DUB6 2/20 0.37
ALOX5 P09917 1/20 0.36
CYP19A1 P11511 1/20 0.34
KCNMA1 Q12791 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27804109 0.85 NOTUM (0.48) CHRNEMAPK1KMT2AHDAC1NOTUM
SCHEMBL4285071 0.84 MAPK1 (0.34) CHRNEHSP90AB1MAPK1KMT2AHDAC1
SCHEMBL2176041 0.75 ALDH1A1 (0.50) MAPK1KMT2A
Hydrochloric Acid SCHEMBL5913639 0.74 ALDH1A1 (0.48) MAPK1KMT2A
SCHEMBL3399659 0.70 MAPT (0.44) MAPK1KMT2A
SCHEMBL15425743 0.69 CYP19A1 (0.67) HSP90AB1CYP19A1
SCHEMBL12432223 0.67 NOTUM (0.42) HSP90AB1NOTUMCYP19A1
SCHEMBL4294198 0.67 KMT2A (0.43) MAPK1KMT2AHDAC1
SCHEMBL16198599 0.67 HDAC1 (0.51) HSP90AB1HDAC1CYP19A1
SCHEMBL1674266 0.66 NOTUM (0.61) NOTUM

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-101981036-B Pyrrolo [2, 3-D] pyridines and use thereof as tyrosine kinase inhibitors NOVARTIS AG 2013-09-04 CN disclosed
CN-101981036-A Pyrrolo [2, 3-D] pyridines and use thereof as tyrosine kinase inhibitors NOVARTIS AG 2011-02-23 CN disclosed