SCHEMBL27804129

SCHEMBL27804129

C[C](C)CN1CCN(Cc2cc(N)ccc2C)C(=O)C1

nearest known ligand 0.60

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPK1 P28482 1/20 0.60
KMT2A Q03164 1/20 0.60
COMT P21964 2/20 0.38
TRPC5 Q9UL62 7/20 0.37
KDM4E B2RXH2 1/20 0.36
ALDH1A1 P00352 1/20 0.36
HPGD P15428 1/20 0.36
HTT P42858 1/20 0.36
ACHE P22303 2/20 0.35
RAD52 P43351 1/20 0.35
BTK Q06187 3/20 0.34
EGFR P00533 1/20 0.34
ERBB2 P04626 1/20 0.34
TEC P42680 1/20 0.34
TXK P42681 1/20 0.34
BLK P51451 1/20 0.34
BMX P51813 1/20 0.34
JAK3 P52333 1/20 0.34
ITK Q08881 1/20 0.34
ERBB4 Q15303 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27804070 0.82 KMT2A (0.49) MAPK1KMT2ACOMTALDH1A1HTT
SCHEMBL28786528 0.81 LMNA (0.45) TRPC5ALDH1A1F10
SCHEMBL27824924 0.77 F10 (0.36) MAPK1KMT2ABTKP2RX7F10
SCHEMBL3396051 0.76 MAPK1 (0.51) MAPK1KMT2ACOMTTRPC5KDM4E
SCHEMBL3398174 0.76 MAPK1 (0.56) MAPK1KMT2ACOMTACHERAD52
SCHEMBL3400888 0.74 KMT2A (0.54) MAPK1KMT2AALDH1A1P2RX7
SCHEMBL27915874 0.74 MAPK1 (0.54) MAPK1KMT2ATRPC5KDM4EALDH1A1
SCHEMBL28237788 0.71 GFER (0.41) KMT2AKDM4EALDH1A1HPGDHTT
SCHEMBL27824915 0.71 NR1H2 (0.46) MAPK1KMT2ACOMTALDH1A1ACHE
SCHEMBL31203025 0.70 MAPK1 (0.52) MAPK1KMT2ATRPC5BTKP2RX7

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-101981036-A Pyrrolo [2, 3-D] pyridines and use thereof as tyrosine kinase inhibitors NOVARTIS AG 2011-02-23 CN disclosed