Formetorex

Formetorex

SCHEMBL2780459

C[C@H](Cc1ccccc1)NC=O

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Full drug profile on Sugi Atlas →

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
TAAR1 Q96RJ0 4/20 1.00
MEN1 O00255 1/20 1.00
KMT2A Q03164 1/20 1.00
EPHX1 P07099 1/20 0.66
SIGMAR1 Q99720 7/20 0.59
SLC18A2 Q05940 1/20 0.59
NPC1 O15118 1/20 0.56
RAB9A P51151 1/20 0.56
CYP3A4 P08684 2/20 0.51
ALDH1A1 P00352 1/20 0.51
HTT P42858 1/20 0.51
CYP2C19 P33261 1/20 0.51
CYP1A2 P05177 1/20 0.50
CYP2D6 P10635 1/20 0.50
TSHR P16473 1/20 0.50

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Formetorex SCHEMBL14944822 1.00 TAAR1 (1.00) TAAR1MEN1KMT2AEPHX1SIGMAR1
Formetorex SCHEMBL1812509 1.00 TAAR1 (1.00) TAAR1MEN1KMT2AEPHX1SIGMAR1
SCHEMBL8763948 0.90 TAAR1 (0.81) TAAR1MEN1KMT2AEPHX1SIGMAR1
SCHEMBL10439420 0.82 KMT2A (0.70) TAAR1MEN1KMT2AEPHX1NPC1
SCHEMBL10439384 0.82 KMT2A (0.70) TAAR1MEN1KMT2AEPHX1NPC1
SCHEMBL14944821 0.82 KMT2A (0.70) TAAR1MEN1KMT2AEPHX1NPC1
SCHEMBL8763940 0.82 TAAR1 (0.69) TAAR1MEN1KMT2AEPHX1SIGMAR1
SCHEMBL11077995 0.81 TAAR1 (0.68) TAAR1MEN1KMT2AEPHX1SIGMAR1
SCHEMBL12280099 0.81 KMT2A (0.68) TAAR1MEN1KMT2AEPHX1SIGMAR1
SCHEMBL11294468 0.81 TAAR1 (0.68) TAAR1MEN1KMT2AEPHX1SIGMAR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 10 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-107892670-B Method for synthesizing formamide derivative through cobalt-catalyzed formylation reaction 湘潭大学 2019-12-13 CN claimed
US-8710268-B2 Method for the hydrolysis of substituted formylamines into substituted amines BOBYLEV MIKHAIL (US) 2014-04-29 US claimed
US-20130046111-A1 Method for the Hydrolysis of Substituted Formylamines into Substituted Amines BOBYLEV MIKHAIL (US) 2013-02-21 US claimed
EP-2175854-A1 IMPROVED METHOD FOR THE SYNTHESIS OF SUBSTITUTED FORMYLAMINES AND SUBSTITUTED AMINES University Of North Dakota Research Foundation (US) 2010-04-21 EP claimed
US-20090143622-A1 Method For The Synthesis Of Substituted Formylamines And Substituted Amines BOBYLEV MIKHAIL 2009-06-04 US claimed
WO-2009018353-A1 IMPROVED METHOD FOR THE SYNTHESIS OF SUBSTITUTED FORMYLAMINES AND SUBSTITUTED AMINES UNIVERSITY OF NORTH DAKOTA RESEARCH FOUNDATION (US) 2009-02-05 WO claimed
EP-1442006-B1 PREPARATION OF AMPHETAMINES FROM PHENYLPROPANOLAMINES BOEHRINGER INGELHEIM CHEMICALS (US) 2005-08-24 EP disclosed
EP-1442006-A2 PREPARATION OF AMPHETAMINES FROM PHENYLPROPANOLAMINES Boehringer Ingelheim Chemicals, Inc. (US) 2004-08-04 EP disclosed
WO-2003037843-A2 PREPARATION OF AMPHETAMINES FROM PHENYLPROPANOLAMINES BOEHRINGER INGELHEIM CHEMICALS, INC. (US) 2003-05-08 WO disclosed
US-6399828-B1 ACYLATION OF PHENYLPROPANOLAMINE; CATALYTIC HYDROGENATION BOEHRINGER INGELHEIM CHEMICALS, INC. 2002-06-04 US disclosed