SCHEMBL11077995

SCHEMBL11077995

C[C@H](Cc1ccccc1)NNC=O

nearest known ligand 0.68

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TAAR1 Q96RJ0 4/20 0.68
MEN1 O00255 1/20 0.68
KMT2A Q03164 1/20 0.68
EPHX1 P07099 1/20 0.56
SIGMAR1 Q99720 7/20 0.55
SLC18A2 Q05940 1/20 0.55
NPC1 O15118 1/20 0.53
RAB9A P51151 1/20 0.53
ADRB2 P07550 1/20 0.49
ADRB1 P08588 1/20 0.49
HTR1A P08908 1/20 0.49
ADORA3 P0DMS8 1/20 0.49
DRD2 P14416 1/20 0.49
ADRA2B P18089 1/20 0.49
ADRA2C P18825 1/20 0.49
CNR1 P21554 1/20 0.49
SLC6A2 P23975 1/20 0.49
HTR2A P28223 1/20 0.49
SLC6A4 P31645 1/20 0.49
MC4R P32245 1/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11294468 1.00 TAAR1 (0.68) TAAR1MEN1KMT2AEPHX1SIGMAR1
SCHEMBL30624762 0.82 SIGMAR1 (0.71) TAAR1MEN1KMT2ASIGMAR1SLC18A2
Formetorex SCHEMBL2780459 0.81 TAAR1 (1.00) TAAR1MEN1KMT2AEPHX1SIGMAR1
Formetorex SCHEMBL14944822 0.81 TAAR1 (1.00) TAAR1MEN1KMT2AEPHX1SIGMAR1
Formetorex SCHEMBL1812509 0.81 TAAR1 (1.00) TAAR1MEN1KMT2AEPHX1SIGMAR1
SCHEMBL27925840 0.75 EPHX1 (0.53) EPHX1CYP1A2
SCHEMBL19285610 0.74 TAAR1 (0.62) TAAR1MEN1KMT2ASIGMAR1SLC18A2
SCHEMBL27884766 0.74 ATM (0.56) RAB9ALMNA
SCHEMBL21243273 0.73 SIGMAR1 (0.73) TAAR1MEN1KMT2ASIGMAR1SLC18A2
SCHEMBL29257172 0.72 EPHX1 (1.00) TAAR1MEN1KMT2AEPHX1SIGMAR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0061907-B1 SECONDARY AMINES, THEIR PREPARATION, PHARMACEUTICAL COMPOSITIONS CONTAINING THEM AND THEIR USE BEECHAM GROUP PLC (GB) 1984-08-01 EP disclosed
EP-0061907-A1 Secondary amines, their preparation, pharmaceutical compositions containing them and their use BEECHAM GROUP PLC (GB) 1982-10-06 EP disclosed