SCHEMBL2781237

SCHEMBL2781237

CN1CCN(CC(NC(=O)OC(C)(C)C)C(=O)O)CC1

nearest known ligand 0.42

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
CTSS P25774 6/20 0.42
CTSK P43235 6/20 0.42
CA1 P00915 1/20 0.41
CA2 P00918 1/20 0.41
CA7 P43166 1/20 0.41
PPARA Q07869 6/20 0.41
PPARG P37231 5/20 0.41
CTSL P07711 1/20 0.40
CTSB P07858 1/20 0.40
ACE P12821 1/20 0.40
PPARD Q03181 2/20 0.39
MAPK1 P28482 1/20 0.39
ITGB3 P05106 2/20 0.38
ITGA2B P08514 2/20 0.38
TSHR P16473 1/20 0.38
IDO1 P14902 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21994715 0.88 CTSK (0.43) CTSSCTSKCA1CA2CA7
SCHEMBL26119172 0.88 CTSK (0.47) CTSSCTSKCA1CA2CA7
SCHEMBL26119175 0.88 CTSK (0.47) CTSSCTSKCA1CA2CA7
SCHEMBL21994717 0.88 CTSK (0.43) CTSSCTSKCA1CA2CA7
SCHEMBL26121197 0.87 CTSK (0.46) CTSSCTSKPPARAPPARGCTSL
SCHEMBL2748877 0.87 CTSK (0.46) CTSSCTSKPPARAPPARGCTSL
SCHEMBL5142788 0.86 CTSK (0.45) CTSSCTSKPPARAPPARGCTSL
SCHEMBL5354771 0.84 ALDH1A1 (0.48) CTSSCTSKPPARAPPARGCTSL
SCHEMBL4360723 0.84 ALDH1A1 (0.48) CTSSCTSKPPARAPPARGCTSL
SCHEMBL5142965 0.83 ALDH1A1 (0.47) CTSSCTSKPPARAPPARGCTSL

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010091104-A1 GLUCOSYLCERAMIDE SYNTHASE INHIBITORS EXELIXIS, INC. (US) 2010-08-12 WO disclosed