SCHEMBL27823934

SCHEMBL27823934

N#CC(N(CC=O)Cc1ccccc1)C(F)(F)F

nearest known ligand 0.41

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.41
GAA P10253 1/20 0.36
TSHR P16473 1/20 0.36
NPBWR1 P48145 1/20 0.36
KMT2A Q03164 1/20 0.36
NPSR1 Q6W5P4 1/20 0.36
MCHR1 Q99705 1/20 0.36
CTSL P07711 5/20 0.35
CYP2C19 P33261 2/20 0.34
KDM4E B2RXH2 1/20 0.33
LMNA P02545 1/20 0.33
CYP1A2 P05177 1/20 0.33
CYP2C9 P11712 1/20 0.33
CA2 P00918 1/20 0.33
SNCA P37840 1/20 0.32
L3MBTL1 Q9Y468 1/20 0.32
CTSS P25774 2/20 0.32
CTSK P43235 1/20 0.32
TDP1 Q9NUW8 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27966619 0.78 KMT2A (0.47) ALDH1A1GAATSHRNPBWR1KMT2A
SCHEMBL195833 0.77 KDM4E (0.39) ALDH1A1TSHRNPSR1CYP2C19KDM4E
SCHEMBL14653906 0.69 ALDH1A1 (0.34) ALDH1A1TSHRKMT2AKDM4ELMNA
SCHEMBL4668886 0.66 ALDH1A1 (0.53) ALDH1A1TSHRKMT2ALMNACA2
SCHEMBL1650495 0.65 CA2 (0.47) ALDH1A1TSHRMCHR1KDM4ECA2
SCHEMBL31390138 0.65 TSHR (0.41) ALDH1A1GAATSHRNPBWR1KMT2A
SCHEMBL27761779 0.64 ALDH1A1 (0.55) ALDH1A1TSHRKMT2ACTSLCYP2C19
SCHEMBL2565075 0.64 ALDH1A1 (0.50) ALDH1A1GAATSHRNPBWR1KMT2A
SCHEMBL40649 0.64 ALDH1A1 (0.45) ALDH1A1TSHRKMT2ACYP2C19CA2
SCHEMBL123966 0.63 CA2 (0.45) ALDH1A1TSHRMCHR1KDM4ECA2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-102333777-B Nitrogen-containing fused heterocyclic compounds and their use as beta-amyloid production inhibitors EISAI R&D MAN CO LTD 2014-06-25 CN disclosed
CN-102333777-A Nitrogen-containing fused heterocyclic compounds and their use as beta-amyloid production inhibitors EISAI R&D MAN CO LTD 2012-01-25 CN disclosed