SCHEMBL27831725

SCHEMBL27831725

C=Cc1nc(C)ccc1OC(C)=O

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PTGS1 P23219 2/20 0.40
SRD5A1 P18405 1/20 0.39
ALDH1A1 P00352 3/20 0.38
TSHR P16473 3/20 0.38
RAB9A P51151 2/20 0.38
KDM4E B2RXH2 2/20 0.38
GAA P10253 1/20 0.38
CFD P00746 1/20 0.37
NR3C1 P04150 1/20 0.36
NPC1 O15118 1/20 0.35
SMN1; SMN2 Q16637 1/20 0.35
MEN1 O00255 1/20 0.35
KMT2A Q03164 1/20 0.35
ALOX5 P09917 1/20 0.35
LMNA P02545 1/20 0.35
ESR1 P03372 1/20 0.35
ITGB3 P05106 1/20 0.35
ITGA2B P08514 1/20 0.35
HMGB1 P09429 1/20 0.35
HPGD P15428 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16742902 0.77 MEN1 (0.54) PTGS1ALDH1A1TSHRRAB9AKDM4E
SCHEMBL4710366 0.75 LMNA (0.42) PTGS1ALDH1A1RAB9AKDM4ENPC1
SCHEMBL4710365 0.75 LMNA (0.42) PTGS1ALDH1A1RAB9AKDM4ENPC1
SCHEMBL4710439 0.74 KMT2A (0.40) ALDH1A1RAB9AKDM4ENPC1SMN1; SMN2
SCHEMBL4710440 0.74 KMT2A (0.40) ALDH1A1RAB9AKDM4ENPC1SMN1; SMN2
SCHEMBL27850348 0.74 CFD (0.44) PTGS1ALDH1A1TSHRRAB9AKDM4E
SCHEMBL27703249 0.74 CFD (0.43) PTGS1ALDH1A1TSHRRAB9AKDM4E
SCHEMBL4710055 0.73 KMT2A (0.44) ALDH1A1RAB9AKDM4EGAANPC1
SCHEMBL4710053 0.73 KMT2A (0.44) ALDH1A1RAB9AKDM4EGAANPC1
SCHEMBL16742712 0.72 KDM4E (0.56) PTGS1ALDH1A1TSHRRAB9AKDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-102300857-A N-{[(ir,4s,6r-3-(2-pyridinylcarbonyl)-3-azabicyclo [4.1.0]hept-4-yl] Methyl}-2-heteroarylamine Derivatives And Uses Thereof 2011-12-28 CN disclosed