SCHEMBL27831797

SCHEMBL27831797

C=CC(=O)Nc1cccc(Nc2ncc(F)c(Nc3ccc(C)cc3)n2)c1

nearest known ligand 0.84

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
EGFR P00533 17/20 0.84
ITK Q08881 9/20 0.84
BTK Q06187 4/20 0.76
JAK2 O60674 1/20 0.73
LYN P07948 1/20 0.73
TEC P42680 1/20 0.73
TXK P42681 1/20 0.73
BMX P51813 1/20 0.73
JAK3 P52333 1/20 0.73
CD69 Q07108 1/20 0.73

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2350864 0.93 EGFR (0.82) EGFRITKBTKJAK2LYN
SCHEMBL29722291 0.92 EGFR (1.00) EGFRITKBTKJAK2LYN
SCHEMBL13165707 0.92 EGFR (1.00) EGFRITKBTKJAK2LYN
SCHEMBL29722526 0.91 EGFR (1.00) EGFRITKBTKJAK2LYN
SCHEMBL13165509 0.91 EGFR (1.00) EGFRITKBTKJAK2LYN
SCHEMBL15815010 0.91 EGFR (0.86) EGFRITKBTKJAK2LYN
SCHEMBL21338060 0.91 EGFR (0.86) EGFRITKBTKJAK2LYN
SCHEMBL28080977 0.89 BTK (0.88) EGFRITKBTKJAK3
SCHEMBL13498409 0.87 EGFR (0.84) EGFRITKBTKJAK2LYN
SCHEMBL28437843 0.87 EGFR (0.77) EGFRITKBTKJAK2LYN

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-102740847-A Heteroaryl compounds and uses thereof AVILA THERAPEUTICS INC 2012-10-17 CN disclosed
CN-102083800-A Heteroaryl compounds and uses thereof AVILA THERAPEUTICS AND USES TH 2011-06-01 CN disclosed